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TargetMol | Compound Library

Bioactive Compound Library

Catalog No. L4000

It contains more than 17520 small molecule compounds, with known biological activities causing biological reaction in cells, tissue even whole body, including Clinical compound library (L3400), Preclinical compound library (L3410), and Approved drug library (L1000). All compounds have clear targets and detailed information description, which is the key point to drug research and development like drug repurposing, small molecule inducing stem cell differentiation, and target identification in mechanism interrogation. Many scientists have identified small molecules that can regulate cell fate and function, and stem cell differentiation by screening annotated bioactive compound library with confirmed activity and known targets. Recent advances in iPSC technology have made reprogramming of somatic cells towards pluripotency possible and simpler. Using both phenotypic screening and hypothesis-driven approaches, a growing number of compounds have been identified that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules with success in cardiomyocyte differentiation and proliferation, neural progenitor cells, etc.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4000

Bioactive Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A collection of 17520 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
  • All compounds have clear targets;
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • Covers various disease research areas, such as Cancer, Metabolism, Immunology and Cardiovascular system, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Antibacterial
Endogenous Metabolite
Autophagy
Antibiotic
5-HT Receptor
AChR
Antifungal
Parasite
Adrenergic Receptor
COX
NF-κB
DNA/RNA Synthesis
Dopamine Receptor
Calcium Channel
CDK
HIV Protease
Potassium Channel
PI3K
Antioxidant
EGFR
Histamine Receptor
Sodium Channel
Dehydrogenase
PDE
Cytochromes P450
Epigenetic Reader Domain
Reactive Oxygen Species
GABA Receptor
VEGFR
GluR
Histone Methyltransferase
PPAR
TRP/TRPV Channel
Influenza Virus
Microtubule Associated
Phosphatase
HDAC
TNF
GPR
Cholinesterase (ChE)
JAK
mTOR
Wnt/beta-catenin
p38 MAPK
Topoisomerase
Akt
SARS-CoV
Prostaglandin Receptor
Src
Estrogen/progestogen Receptor
Antiviral
ERK
PKC
RAAS
Adenosine Receptor
FLT
Ferroptosis
Opioid Receptor
IL Receptor
HCV Protease
STAT
PARP
NMDAR
Estrogen Receptor/ERR
PDGFR
iGluR
Nucleoside Antimetabolite/Analog
MMP
AMPK
Caspase
GSK-3
FGFR
Bcl-2 Family
NO Synthase
Virus Protease
Raf
Lipoxygenase
MAO
Glucocorticoid Receptor
Androgen Receptor
TLR
c-Kit
c-Met/HGFR
Beta Amyloid
Cannabinoid Receptor
ATPase
HBV
ROS
Phospholipase
Bcr-Abl
HSP
Proteasome
TGF-beta/Smad
ALK
Mitochondrial Metabolism
HSV
Anti-infection
Tyrosinase
Sirtuin
Drug Metabolite
BTK
Nrf2
ADC Cytotoxin
Histone Demethylase
MAPK
DUB
Integrin
Antifection
HIF/HIF Prolyl-Hydroxylase
NOS
JNK
Ras
Aurora Kinase
PKA
P-gp
Kras
HER
Tyrosine Kinases
Transferase
Mitophagy
ROCK
E1/E2/E3 Enzyme
CCR
p53
Gamma-secretase
IκB/IKK
MEK
Monoamine Oxidase
Carbonic Anhydrase
Immunology/Inflammation related
Interleukin
Reverse Transcriptase
Casein Kinase
HIF
Neurokinin receptor
Serotonin Transporter
P2X Receptor
CXCR
Retinoid Receptor
Reductase
Cysteine Protease
Norepinephrine
Serine/threonin kinase
S1P Receptor
PROTACs
Serine Protease
IGF-1R
Glucosidase
DNA-PK
FAK
Hedgehog/Smoothened
CaMK
c-RET
NOD
LPL Receptor
Histone Acetyltransferase
TAM Receptor
RIP kinase
Trk receptor
Sigma receptor
FAAH
Proton pump
transporter
S6 Kinase
Chloride channel
Progesterone Receptor
Glucokinase
Fatty Acid Synthase
PLK
Amino Acids and Derivatives
PERK
Acyltransferase
ATM/ATR
c-Fms
ribosome
CFTR
DPP-4
Syk
HMG-CoA Reductase
Thrombin
Mdm2
Neuropeptide Y Receptor
Endothelin Receptor
Protease-activated Receptor
Chk
DNA
Thyroid hormone receptor(THR)
NADPH
Rho
Pim
Aryl Hydrocarbon Receptor
Glucagon Receptor
cAMP
AhR
Kinesin
Smo
Complement System
DNA Methyltransferase
IRAK
ROR
P2Y Receptor
LTR
BACE
Lipase
Factor Xa
Leukotriene Receptor
STING
Melanocortin Receptor
cholecystokinin
PD-1/PD-L1
DHFR
DNA Alkylator/Crosslinker
FXR
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
LPA Receptor
PDK
DYRK
Guanylate cyclase
Platelet aggregation
Glutathione Peroxidase
MRP
Bradykinin Receptor
OX Receptor
Xanthine Oxidase
Epoxide Hydrolase
LRRK2
Hydroxylase
YAP
Vasopressin Receptor
Ligand for E3 Ligase
c-Myc
GNRH Receptor
DNA Alkylation
PAK
RSV
Aromatase
GTPase
Liver X Receptor
IAP
Ephrin Receptor
ROS Kinase
NOD-like Receptor (NLR)
IRE1
Myosin
PGE Synthase
PI4K
Antifolate
ABC Transporter
Telomerase
GHSR
Neurotensin Receptor
CSF-1R
LDL
Somatostatin
Lipid
Beta-Secretase
Aminopeptidase
NADPH-oxidase
Monocarboxylate transporter
DNA gyrase
GPCR19
PAI-1
CaSR
Vitamin
Glutaminase
PAFR
Phosphorylase
Monoamine Transporter
Stearoyl-CoA Desaturase (SCD)
Acetyl-CoA Carboxylase
Discoidin Domain Receptor (DDR)
Ligands for Target Protein for PROTAC
IFNAR
Arrestin
CETP
NAMPT
IDO
GRK
Isocitrate Dehydrogenase (IDH)
Free radical scavengers
GST
PKM
Melatonin Receptor
UGT
Molecular Glues
Bombesin Receptor
BCRP
MNK
OAT
GPX
Imidazoline Receptor
Adenylyl Cyclase
Dynamin
LIM Kinase
MT Receptor
ATP Citrate Lyase
Wee1
PSMA
Porcupine
Neprilysin
Gap Junction Protein
MLK
Apelin receptor
Arginase
Tie-2
SIK
GlyT
Angiotensin-converting Enzyme (ACE)
PTEN
PAD
ASK
SGK
Melanin-concentrating Hormone Receptor (MCHR)
CRM1
Na+/Ca2+ Exchanger
OCT
AAK1
PYK2
Amylase
Annexin A
MAGL
cGAS
CRFR
Methionine Adenosyltransferase (MAT)
Carboxypeptidase
Protease
Oxytocin Receptor
CGRP Receptor
APC/C
p97
MALT
MyD88
RAR/RXR 
Cell wall
FLAP
Transketolase
Survivin
Decarboxylase
ADC Linker
TSH Receptor
Pyroptosis
MELK
CRISPR/Cas9
Adenosine Deaminase
DAPK
Glyoxalase
DprE1
VDAC
Cell Cycle Arrest
MTH1
PROTAC Linker
HCN Channel
ACK1
MRGPR
CD73
Hippo pathway
Aquaporin
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
NEDD8
gp120/CD4
TOPK
Galectin
Kisspeptin
Hck
RANKL/RANK
Adiponectin Receptor
Hexokinase
KSP
Thrombopoietin Receptor
AIM2
IGF-2R
Transaminase
Necroptosis
Haspin Kinase
FABP
Na-K-Cl cotransporter
Mucin
OXPHOS
Glutathione reductase
CPT
GluCls
HuR
KLF
Cuproptosis
Taste receptor
GSNOR
Piezo Channel
NUDIX hydrolase
EBI2/GPR183
Sodium-dependent phosphate transporter
Glutaminyl Cyclase
VDA
FOXO1
Prolyl Endopeptidase (PREP)
Fas/FasL
PACAP
Integrase
PGC-1α
hCE
RXFP receptor
ATTECs
Lysosomal Autophagy
Liposome
LYTACs
stilbene oxidase
CYP19A1
Procollagen C Proteinase
Neuropeptide W
Aconitase
LHRH
N-Acetylglucosaminyltransferase
Stemness kinase
Motilin Receptor
Anion Exchanger
Thioredoxin
Huntingtin
FKBP
Fer/FerT kinase
NMU2R