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TargetMol | Compound Library

Bioactive Compound Library

Catalog No. L4000

It contains more than 17100 small molecule compounds, with known biological activities causing biological reaction in cells, tissue even whole body, including Clinical compound library (L3400), Preclinical compound library (L3410), and Approved drug library (L1000). All compounds have clear targets and detailed information description, which is the key point to drug research and development like drug repurposing, small molecule inducing stem cell differentiation, and target identification in mechanism interrogation. Many scientists have identified small molecules that can regulate cell fate and function, and stem cell differentiation by screening annotated bioactive compound library with confirmed activity and known targets. Recent advances in iPSC technology have made reprogramming of somatic cells towards pluripotency possible and simpler. Using both phenotypic screening and hypothesis-driven approaches, a growing number of compounds have been identified that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules with success in cardiomyocyte differentiation and proliferation, neural progenitor cells, etc.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L4000

Bioactive Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A collection of 17100 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
  • All compounds have clear targets;
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • Covers various disease research areas, such as Cancer, Metabolism, Immunology and Cardiovascular system, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Antibacterial
Endogenous Metabolite
Autophagy
Antibiotic
5-HT Receptor
AChR
Antifungal
Parasite
Adrenergic Receptor
COX
NF-κB
DNA/RNA Synthesis
Dopamine Receptor
Calcium Channel
CDK
HIV Protease
Potassium Channel
PI3K
EGFR
Antioxidant
Histamine Receptor
PDE
P450
Epigenetic Reader Domain
Dehydrogenase
Sodium Channel
Reactive Oxygen Species
GABA Receptor
VEGFR
GluR
JAK
Histone Methyltransferase
PPAR
Influenza Virus
TRP/TRPV Channel
Microtubule Associated
HDAC
TNF
GPR
Phosphatase
AChE
Wnt/beta-catenin
mTOR
Akt
Topoisomerase
p38 MAPK
Prostaglandin Receptor
Estrogen/progestogen Receptor
SARS-CoV
PKC
ERK
Antiviral
Src
Adenosine Receptor
FLT
Ferroptosis
IL Receptor
HCV Protease
RAAS
PARP
Opioid Receptor
STAT
NMDAR
Estrogen Receptor/ERR
PDGFR
Caspase
iGluR
Nucleoside Antimetabolite/Analog
AMPK
GSK-3
MMP
NO Synthase
FGFR
Raf
Virus Protease
BCL
Lipoxygenase
MAO
Androgen Receptor
c-Kit
Glucocorticoid Receptor
Beta Amyloid
Phospholipase
Bcr-Abl
c-Met/HGFR
HBV
TLR
Cannabinoid Receptor
ATPase
ROS
Proteasome
HSP
TGF-beta/Smad
Mitochondrial Metabolism
ALK
HSV
Sirtuin
Anti-infection
Tyrosinase
CCR
Drug Metabolite
BTK
MAPK
JNK
Histone Demethylase
Antifection
DUB
HIF/HIF Prolyl-Hydroxylase
NOS
Integrin
Aurora Kinase
Nrf2
PKA
HER
ADC Cytotoxin
Kras
Ras
Mitophagy
Tyrosine Kinases
E1/E2/E3 Enzyme
P-gp
Transferase
ROCK
p53
IκB/IKK
Monoamine Oxidase
Carbonic Anhydrase
MEK
Immunology/Inflammation related
Gamma-secretase
Interleukin
Casein Kinase
Reverse Transcriptase
HIF
Neurokinin receptor
Serotonin Transporter
CXCR
Cysteine Protease
Retinoid Receptor
Reductase
Serine/threonin kinase
P2X Receptor
Norepinephrine
S1P Receptor
IGF-1R
Serine Protease
Glucosidase
DNA-PK
Hedgehog/Smoothened
CaMK
c-RET
Trk receptor
Histone Acetyltransferase
NOD
FAK
LPL Receptor
RIP kinase
TAM Receptor
PROTACs
FAAH
Sigma receptor
Proton pump
S6 Kinase
Chloride channel
Glucokinase
Acyltransferase
transporter
Amino Acids and Derivatives
Progesterone Receptor
Fatty Acid Synthase
ATM/ATR
c-Fms
ribosome
PLK
Mdm2
Syk
Thrombin
CFTR
PERK
Neuropeptide Y Receptor
Endothelin Receptor
HMG-CoA Reductase
NADPH
DPP-4
Chk
Protease-activated Receptor
Rho
Thyroid hormone receptor(THR)
Pim
Aryl Hydrocarbon Receptor
Glucagon Receptor
cAMP
DNA Methyltransferase
Smo
DNA
Complement System
IRAK
AhR
Kinesin
DHFR
ROR
DNA Alkylator/Crosslinker
BACE
Lipase
FXR
cholecystokinin
P2Y Receptor
LTR
Factor Xa
Leukotriene Receptor
Guanylate cyclase
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
STING
LPA Receptor
PDK
PD-1/PD-L1
DYRK
LRRK2
Glutathione Peroxidase
MRP
DNA Alkylation
Bradykinin Receptor
Xanthine Oxidase
Epoxide Hydrolase
Melanocortin Receptor
Hydroxylase
Platelet aggregation
OX Receptor
YAP
c-Myc
GNRH Receptor
IAP
PAK
Vasopressin Receptor
RSV
Aromatase
GTPase
Liver X Receptor
IRE1
Myosin
Ephrin Receptor
PI4K
ROS Kinase
NOD-like Receptor (NLR)
ABC
Antifolate
Telomerase
PGE Synthase
GHSR
Neurotensin Receptor
CSF-1R
LDL
Somatostatin
Lipid
Beta-Secretase
Aminopeptidase
Monocarboxylate transporter
DNA gyrase
Monoamine Transporter
GPCR19
NADPH-oxidase
CaSR
Phosphorylase
Stearoyl-CoA Desaturase (SCD)
PAI-1
Acetyl-CoA Carboxylase
Discoidin Domain Receptor (DDR)
Arrestin
CETP
NAMPT
Glutaminase
IDO
PAFR
GRK
Isocitrate Dehydrogenase (IDH)
Free radical scavengers
GST
PKM
IFNAR
Vitamin
UGT
Bombesin Receptor
BCRP
GPX
MLK
Imidazoline Receptor
Adenylyl cyclase
Dynamin
Ligands for Target Protein for PROTAC
Melatonin Receptor
LIM Kinase
MT Receptor
ATP Citrate Lyase
PSMA
MNK
OAT
Neprilysin
SGK
Gap Junction Protein
CAT
Arginase
Tie-2
SIK
GlyT
Angiotensin-converting Enzyme (ACE)
PTEN
PAD
Porcupine
ASK
Ligand for E3 Ligase
Apelin receptor
CRM1
Na+/Ca2+ Exchanger
OCT
Amylase
Annexin A
AAK1 (AP2 associated kinase 1)
Molecular Glues
APC
MAGL
Wee1
cGAS
CRFR
Carboxypeptidase
Protease
Oxytocin Receptor
p97
Melanin-concentrating Hormone Receptor (MCHR)
MyD88
RAR/RXR 
Cell wall
PYK2
FLAP
Transketolase
Survivin
Decarboxylase
TSH Receptor
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
CRISPR/Cas9
Adenosine deaminase
CGRP Receptor
DAPK
MALT
DprE1
TOPK
Galectin
VDAC
cell cycle arrest
MTH1
HCN Channel
ACK
MRGPR
CD73
Hippo pathway
Aquaporin
BMI-1
advanced glycation end products
NPC1L1
CD38
NEDD8
gp120/CD4
Kisspeptin
Adiponectin receptor
Hexokinase
KSP
Thrombopoietin Receptor
AIM2
Transaminase
Necroptosis
Hck
RANKL/RANK
Haspin Kinase
Na-K-Cl cotransporter
Mucin
OXPHOS
Glutathione reductase
CPT
GluCls
HuR
KLF
Cuproptosis
Glyoxalase
Taste receptor
GSNOR
NUDIX hydrolase
Piezo Channel
EBI2/GPR183
VDA
FOXO1
Prolyl Endopeptidase (PREP)
Fas/FasL
PACAP
Integrase
PGC-1α
hCE
RXFP receptor
ATTECs
IGF-2R
lysosomal autophagy
Liposome
LYTACs
stilbene oxidase
CYP19A1
Procollagen C Proteinase
aconitase
Neuropeptide W
LHRH
N-Acetylglucosaminyltransferase
Stemness kinase
FABP
Anion Exchanger
Thioredoxin
Fer/FerT kinase
NMU2R