Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Bioactive Compound Library

Catalog No. L4000

It contains more than 17760 small molecule compounds, with known biological activities causing biological reaction in cells, tissue even whole body, including Clinical compound library (L3400), Preclinical compound library (L3410), and Approved drug library (L1000). All compounds have clear targets and detailed information description, which is the key point to drug research and development like drug repurposing, small molecule inducing stem cell differentiation, and target identification in mechanism interrogation.

Many scientists have identified small molecules that can regulate cell fate and function, and stem cell differentiation by screening annotated bioactive compound library with confirmed activity and known targets. Recent advances in iPSC technology have made reprogramming of somatic cells towards pluripotency possible and simpler. Using both phenotypic screening and hypothesis-driven approaches, a growing number of compounds have been identified that can functionally replace reprogramming transcription factors, enhance efficiency of iPSC generation and accelerate the reprogramming process by single use or a combination of several molecules with success in cardiomyocyte differentiation and proliferation, neural progenitor cells, etc.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L4000

Bioactive Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A collection of 17760 small molecule compounds with validated activity for high throughput screening (HTS), high content screening (HCS), cell induction, and target identification;
  • All compounds have clear targets;
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • Covers various disease research areas, such as Cancer, Metabolism, Immunology and Cardiovascular system, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Apoptosis
Antibacterial
Endogenous Metabolite
Autophagy
Antibiotic
5-HT Receptor
AChR
Antifungal
Parasite
Adrenergic Receptor
COX
NF-κB
DNA/RNA Synthesis
Dopamine Receptor
Calcium Channel
CDK
HIV Protease
Potassium Channel
Antioxidant
PI3K
EGFR
Histamine Receptor
Epigenetic Reader Domain
Sodium Channel
Cytochromes P450
Dehydrogenase
PDE
Reactive Oxygen Species
GABA Receptor
VEGFR
GluR
Histone Methyltransferase
PPAR
TRP/TRPV Channel
Influenza Virus
Microtubule Associated
HDAC
TNF
Phosphatase
GPR
Cholinesterase (ChE)
Wnt/beta-catenin
JAK
mTOR
Topoisomerase
Akt
p38 MAPK
SARS-CoV
Prostaglandin Receptor
Antiviral
Estrogen/progestogen Receptor
Src
ERK
RAAS
PKC
Ferroptosis
PARP
Adenosine Receptor
IL Receptor
STAT
FLT
HCV Protease
NMDAR
Opioid Receptor
Estrogen Receptor/ERR
Nucleoside Antimetabolite/Analog
iGluR
PDGFR
Caspase
MMP
AMPK
FGFR
GSK-3
Virus Protease
Bcl-2 Family
NO Synthase
Raf
Lipoxygenase
Glucocorticoid Receptor
TLR
MAO
Androgen Receptor
c-Kit
ROS
Beta Amyloid
c-Met/HGFR
HBV
HSP
Phospholipase
Cannabinoid Receptor
ATPase
Bcr-Abl
Proteasome
ALK
TGF-beta/Smad
Mitochondrial Metabolism
HSV
Anti-infection
Tyrosinase
Drug Metabolite
MAPK
Sirtuin
Nrf2
Histone Demethylase
JNK
DUB
HIF/HIF Prolyl-Hydroxylase
Integrin
Antifection
NOS
PKA
Ras
Aurora Kinase
HER
Transferase
E1/E2/E3 Enzyme
Mitophagy
Tyrosine Kinases
ROCK
CCR
P-gp
p53
Gamma-secretase
IκB/IKK
Monoamine Oxidase
Carbonic Anhydrase
Immunology/Inflammation related
Casein Kinase
MEK
Neurokinin receptor
Interleukin
Reverse Transcriptase
HIF
Cysteine Protease
P2X Receptor
CXCR
S1P Receptor
Reductase
Retinoid Receptor
Serotonin Transporter
Norepinephrine
PROTACs
Serine Protease
Serine/threonin kinase
Glucosidase
IGF-1R
FAK
CaMK
DNA-PK
LPL Receptor
RIP kinase
Hedgehog/Smoothened
c-RET
NOD
Histone Acetyltransferase
TAM Receptor
Trk receptor
Sigma receptor
S6 Kinase
FAAH
Proton pump
Fatty Acid Synthase
transporter
ATM/ATR
Chloride channel
PERK
Progesterone Receptor
Glucokinase
c-Fms
PLK
Amino Acids and Derivatives
Acyltransferase
ribosome
CFTR
Mdm2
DPP-4
Syk
HMG-CoA Reductase
Pim
Neuropeptide Y Receptor
Endothelin Receptor
Thrombin
Protease-activated Receptor
NADPH
Chk
DNA
Cholecystokinin Receptor
Rho
DNA Methyltransferase
Kinesin
Thyroid hormone receptor(THR)
Aryl Hydrocarbon Receptor
Glucagon Receptor
cAMP
AhR
DHFR
LTR
Smo
STING
Complement System
IRAK
ROR
P2Y Receptor
BACE
Lipase
Leukotriene Receptor
FXR
LPA Receptor
Melanocortin Receptor
PDK
DNA Alkylator/Crosslinker
DYRK
Factor Xa
Guanylate cyclase
Xanthine Oxidase
Indoleamine 2,3-Dioxygenase (IDO)
SGLT
PD-1/PD-L1
BTK
ADC Cytotoxin
Glutathione Peroxidase
MRP
LRRK2
Platelet aggregation
YAP
Bradykinin Receptor
Vasopressin Receptor
OX Receptor
Epoxide Hydrolase
Hydroxylase
c-Myc
GNRH Receptor
Kras
Liver X Receptor
DNA Alkylation
PAK
Ephrin Receptor
RSV
Aromatase
GTPase
IAP
ROS Kinase
NOD-like Receptor (NLR)
Antifolate
Myosin
IRE1
PGE Synthase
Ligand for E3 Ligase
PI4K
ABC Transporter
Telomerase
GHSR
Neurotensin Receptor
CSF-1R
LDL
Somatostatin
Lipid
Beta-Secretase
Aminopeptidase
NADPH-oxidase
Monocarboxylate transporter
Molecular Glues
GPCR19
PAI-1
Acetyl-CoA Carboxylase
MicroRNA
Arrestin
Glutaminase
PAFR
DNA gyrase
Monoamine Transporter
Stearoyl-CoA Desaturase (SCD)
Discoidin Domain Receptor (DDR)
Ligands for Target Protein for PROTAC
IFNAR
CETP
CaSR
NAMPT
IDO
GRK
Phosphorylase
Isocitrate Dehydrogenase (IDH)
MNK
Free radical scavengers
GPX
PKM
Apelin receptor
Melatonin Receptor
UGT
Bombesin Receptor
BCRP
OAT
GST
Imidazoline Receptor
Adenylyl Cyclase
Dynamin
Arginase
Tie-2
LIM Kinase
MT Receptor
Angiotensin-converting Enzyme (ACE)
ATP Citrate Lyase
Porcupine
Neprilysin
Gap Junction Protein
MLK
GlyT
PTEN
PAD
Wee1
ASK
SGK
APC/C
Melanin-concentrating Hormone Receptor (MCHR)
CRM1
Na+/Ca2+ Exchanger
OCT
AAK1
PYK2
Amylase
SIK
Annexin A
MAGL
cGAS
CRFR
TSH Receptor
Methionine Adenosyltransferase (MAT)
Carboxypeptidase
Protease
Oxytocin Receptor
CGRP Receptor
p97
RAR/RXR
MALT
MyD88
FLAP
HCN Channel
Survivin
Decarboxylase
Pyroptosis
MELK
CRISPR/Cas9
Adenosine Deaminase
DAPK
NEDD8
DprE1
Cell wall
VDAC
Hck
Cell Cycle Arrest
MTH1
ACK1
MRGPR
CD73
Hippo pathway
Aquaporin
BMI-1
Advanced Glycation End Products
NPC1L1
CD38
gp120/CD4
TOPK
Galectin
Kisspeptin
Vitamin
RANKL/RANK
Adiponectin Receptor
Hexokinase
KSP
Thrombopoietin Receptor
AIM2
Transaminase
Necroptosis
Haspin Kinase
FABP
Na-K-Cl cotransporter
OXPHOS
PSMA
Glutathione reductase
CPT
GluCls
HuR
KLF
Liposome
Taste receptor
GSNOR
NUDIX hydrolase
Piezo Channel
EBI2/GPR183
Glutaminyl Cyclase
VDA
FOXO1
Prolyl Endopeptidase (PREP)
Fas/FasL
PACAP
Integrase
PROTAC Linker
Transketolase
ADC Linker
hCE
RXFP receptor
ATTECs
Lysosomal Autophagy
Glyoxalase
IGF-2R
stilbene oxidase
CYP19A1
Procollagen C Proteinase
Aconitase
Neuropeptide W
LHRH
N-Acetylglucosaminyltransferase
Stemness kinase
Motilin Receptor
Anion Exchanger
Thioredoxin
glycosidase
Mucin
Huntingtin
FKBP
Cuproptosis
REV-ERB
Fer/FerT kinase
NMU2R
Sodium-dependent phosphate transporter
PGC-1α