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TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3404 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence. Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
HIV Protease
AChR
Dopamine Receptor
COX
Histamine Receptor
VEGFR
Parasite
Sodium Channel
Calcium Channel
EGFR
Antifungal
PI3K
Potassium Channel
PDE
Topoisomerase
FLT
HCV Protease
CDK
Cytochromes P450
PDGFR
Dehydrogenase
JAK
Microtubule Associated
Reactive Oxygen Species
SARS-CoV
PPAR
FGFR
c-Kit
Glucocorticoid Receptor
mTOR
Ferroptosis
Influenza Virus
HDAC
c-Met/HGFR
Src
Estrogen/progestogen Receptor
GABA Receptor
RAAS
HBV
NF-κB
Mitophagy
Prostaglandin Receptor
Reverse Transcriptase
Nucleoside Antimetabolite/Analog
GPR
Adenosine Receptor
Tyrosine Kinases
Raf
Bcr-Abl
BTK
Proteasome
Androgen Receptor
Serotonin Transporter
iGluR
Epigenetic Reader Domain
ADC Cytotoxin
Aurora Kinase
Akt
Phosphatase
Virus Protease
TRP/TRPV Channel
ROS
HSV
HER
Transferase
p38 MAPK
Progesterone Receptor
Estrogen Receptor/ERR
PARP
GluR
Norepinephrine
Opioid Receptor
Beta Amyloid
MEK
NMDAR
IL Receptor
HSP
ALK
c-RET
TNF
HIF/HIF Prolyl-Hydroxylase
ATPase
DPP-4
P-gp
Trk receptor
Carbonic Anhydrase
Antioxidant
Antifection
Cholinesterase (ChE)
Antiviral
Histone Methyltransferase
GSK-3
ERK
CXCR
c-Fms
ribosome
Thrombin
DNA Alkylator/Crosslinker
PKC
Gamma-secretase
Mitochondrial Metabolism
Endothelin Receptor
Interleukin
TLR
Retinoid Receptor
Proton pump
MAO
CCR
MMP
Chk
Bcl-2 Family
Phospholipase
S1P Receptor
Thyroid hormone receptor(THR)
DNA-PK
LPL Receptor
E1/E2/E3 Enzyme
SGLT
STAT
AMPK
HIF
Syk
CFTR
p53
NO Synthase
Caspase
Guanylate cyclase
TAM Receptor
Integrin
NADPH
Wnt/beta-catenin
Antifolate
CSF-1R
DNA Alkylation
Hedgehog/Smoothened
IGF-1R
Nrf2
Neurokinin receptor
Mdm2
CETP
Glutathione Peroxidase
MRP
PKA
P2X Receptor
Lipoxygenase
TGF-beta/Smad
Hydroxylase
PLK
Cannabinoid Receptor
FAK
Monoamine Oxidase
P2Y Receptor
Reductase
GNRH Receptor
ROCK
IAP
Drug Metabolite
Glucosidase
Vasopressin Receptor
Indoleamine 2,3-Dioxygenase (IDO)
RSV
ATM/ATR
Kras
HMG-CoA Reductase
S6 Kinase
ROS Kinase
DHFR
Histone Demethylase
JNK
Serine Protease
FXR
Aryl Hydrocarbon Receptor
RIP kinase
Smo
OX Receptor
Xanthine Oxidase
DNA
Beta-Secretase
Aminopeptidase
Sirtuin
Casein Kinase
Sigma receptor
Kinesin
ROR
Amino Acids and Derivatives
BACE
Pim
Leukotriene Receptor
Glucokinase
Glucagon Receptor
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
IκB/IKK
DNA Methyltransferase
IRAK
AhR
Tie-2
Factor Xa
IDO
DNA gyrase
Fatty Acid Synthase
Acyltransferase
Ephrin Receptor
Ligand for E3 Ligase
Complement System
Chloride channel
NOS
DprE1
YAP
LTR
IFNAR
Melatonin Receptor
Liver X Receptor
MT Receptor
Monoamine Transporter
Molecular Glues
Neuropeptide Y Receptor
FAAH
KSP
CaMK
Wee1
PGE Synthase
Decarboxylase
CRFR
Neprilysin
Acetyl-CoA Carboxylase
Melanocortin Receptor
GHSR
CGRP Receptor
Gap Junction Protein
NADPH-oxidase
cholecystokinin
CRM1
Arginase
Cell wall
PERK
CaSR
Rho
Serine/threonin kinase
Cysteine Protease
NAMPT
Myosin
Annexin A
ABC Transporter
GlyT
Somatostatin
DUB
Telomerase
PSMA
MAPK
OAT
STING
Free radical scavengers
GPCR19
LPA Receptor
PDK
Adenosine Deaminase
Ras
Tyrosinase
Protease-activated Receptor
NOD-like Receptor (NLR)
Imidazoline Receptor
PD-1/PD-L1
Taste receptor
PROTACs
GSNOR
NEDD8
Ligands for Target Protein for PROTAC
VDA
Galectin
Vitamin
PYK2
IRE1
UGT
LDL
Na-K-Cl cotransporter
Hexokinase
Integrase
HCN Channel
Stearoyl-CoA Desaturase (SCD)
Epoxide Hydrolase
ATP Citrate Lyase
BCRP
Porcupine
CD73
transporter
PAI-1
Drug-Linker Conjugates for ADC
GST
Oxytocin Receptor
Discoidin Domain Receptor (DDR)
p97
MLK
Advanced Glycation End Products
Adenylyl Cyclase
Monocarboxylate transporter
NPC1L1
Hydrogenase
MALT
Arrestin
RAR/RXR 
DYRK
Lipase
GTPase
c-Myc
N-Acetylglucosaminyltransferase
AAK1
VDAC
Hck
Stemness kinase
Glutaminase
FLAP
PAFR
Fas/FasL
GRK
Phosphorylase
Anion Exchanger
PROTAC Linker
Thioredoxin
ACK1
Lipid
MNK
Survivin
Histone Acetyltransferase
ASK
GluCls
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
Aromatase
KLF
PI4K
CRISPR/Cas9
Aquaporin
SGK
Anti-infection
BMI-1
NOD
PKM