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TargetMol | Compound Library

Clinical Compound Library

Catalog No. L3400

Clinical compound library is a collection of 3404 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence. Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L3400

Clinical Compound Library
sizeIn stock
  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3404 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
Endogenous Metabolite
5-HT Receptor
Adrenergic Receptor
DNA/RNA Synthesis
HIV Protease
AChR
Dopamine Receptor
COX
VEGFR
Histamine Receptor
Parasite
Sodium Channel
Calcium Channel
EGFR
PI3K
Antifungal
Potassium Channel
PDE
FLT
Topoisomerase
CDK
HCV Protease
PDGFR
P450
JAK
c-Kit
Dehydrogenase
PPAR
Reactive Oxygen Species
FGFR
Microtubule Associated
SARS-CoV
Ferroptosis
HDAC
Glucocorticoid Receptor
mTOR
c-Met/HGFR
Influenza Virus
Estrogen/progestogen Receptor
Src
Mitophagy
NF-κB
RAAS
Prostaglandin Receptor
GABA Receptor
HBV
Nucleoside Antimetabolite/Analog
Reverse Transcriptase
Tyrosine Kinases
GPR
Adenosine Receptor
Bcr-Abl
Proteasome
Raf
BTK
Androgen Receptor
PARP
Serotonin Transporter
iGluR
Akt
HER
Aurora Kinase
Epigenetic Reader Domain
Virus Protease
ROS
Opioid Receptor
HSV
MEK
Transferase
Norepinephrine
Phosphatase
Progesterone Receptor
Estrogen Receptor/ERR
IL Receptor
GluR
HSP
p38 MAPK
ALK
Beta Amyloid
c-RET
TNF
HIF/HIF Prolyl-Hydroxylase
ERK
Antifection
DPP-4
P-gp
Trk receptor
ATPase
Carbonic Anhydrase
Antioxidant
DNA Alkylator/Crosslinker
TRP/TRPV Channel
NMDAR
ribosome
GSK-3
PKC
AChE
c-Fms
Thrombin
Proton pump
Gamma-secretase
Mitochondrial Metabolism
CXCR
Endothelin Receptor
Interleukin
TLR
Retinoid Receptor
TAM Receptor
DNA-PK
MAO
E1/E2/E3 Enzyme
BCL
CCR
MMP
Chk
Antiviral
STAT
AMPK
Phospholipase
Histone Methyltransferase
LPL Receptor
Caspase
SGLT
HIF
Syk
NO Synthase
S1P Receptor
Thyroid hormone receptor(THR)
Antifolate
Guanylate cyclase
DNA Alkylation
CFTR
p53
Integrin
NADPH
CSF-1R
Hedgehog/Smoothened
IGF-1R
Nrf2
CETP
Glutathione Peroxidase
MRP
PKA
Wnt/beta-catenin
P2X Receptor
Lipoxygenase
TGF-beta/Smad
Hydroxylase
PLK
Cannabinoid Receptor
HMG-CoA Reductase
S6 Kinase
FAK
Monoamine Oxidase
DHFR
P2Y Receptor
Reductase
JNK
GNRH Receptor
ROCK
IAP
Drug Metabolite
Glucosidase
Vasopressin Receptor
OX Receptor
Indoleamine 2,3-Dioxygenase (IDO)
Sirtuin
Casein Kinase
ATM/ATR
Neurokinin receptor
Ras
ROS Kinase
Mdm2
CAT
Histone Demethylase
Pim
Serine Protease
FXR
Aryl Hydrocarbon Receptor
Smo
Xanthine Oxidase
Beta-Secretase
Aminopeptidase
RSV
DNA Methyltransferase
Sigma receptor
Kinesin
ROR
Amino Acids and Derivatives
BACE
Glucokinase
RIP kinase
Isocitrate Dehydrogenase (IDH)
PAK
Bradykinin Receptor
DNA
IκB/IKK
Ligand for E3 Ligase
IRAK
AhR
Tie-2
Factor Xa
Leukotriene Receptor
IDO
Glucagon Receptor
DNA gyrase
Fatty Acid Synthase
Acyltransferase
Ephrin Receptor
Complement System
Chloride channel
NOS
DprE1
LTR
IFNAR
Melatonin Receptor
Liver X Receptor
MT Receptor
Monoamine Transporter
Molecular Glues
FAAH
KSP
CaMK
Wee1
PGE Synthase
Decarboxylase
CRFR
Neprilysin
Acetyl-CoA Carboxylase
GHSR
CGRP Receptor
Gap Junction Protein
NADPH-oxidase
cholecystokinin
CRM1
Arginase
YAP
Cell wall
ABC
CaSR
Rho
Serine/threonin kinase
Cysteine Protease
NAMPT
Myosin
Annexin A
GlyT
Neuropeptide Y Receptor
Somatostatin
DUB
Telomerase
OAT
STING
Free radical scavengers
GPCR19
LPA Receptor
Melanocortin Receptor
PDK
Adenosine deaminase
Tyrosinase
Protease-activated Receptor
NOD-like Receptor (NLR)
Imidazoline Receptor
PD-1/PD-L1
Taste receptor
NEDD8
Ligands for Target Protein for PROTAC
PERK
VDA
Galectin
PYK2
IRE1
UGT
LDL
Na-K-Cl cotransporter
Hexokinase
Integrase
Stearoyl-CoA Desaturase (SCD)
Epoxide Hydrolase
ATP Citrate Lyase
Lipid
BCRP
MAPK
Porcupine
CD73
transporter
PAI-1
GST
Oxytocin Receptor
Discoidin Domain Receptor (DDR)
p97
MLK
advanced glycation end products
Adenylyl cyclase
PROTACs
GSNOR
NPC1L1
Monocarboxylate transporter
Hydrogenase
MALT
Arrestin
RAR/RXR 
DYRK
Lipase
TOPK
GTPase
c-Myc
N-Acetylglucosaminyltransferase
VDAC
Hck
Stemness kinase
Glutaminase
FLAP
Motilin Receptor
PAFR
MTH1
Fas/FasL
GRK
Phosphorylase
AAK1 (AP2 associated kinase 1)
Anion Exchanger
PROTAC Linker
HCN Channel
Thioredoxin
ACK
MNK
Survivin
Histone Acetyltransferase
ASK
GluCls
Pyroptosis
MELK
Methionine Adenosyltransferase (MAT)
Hippo pathway
Aromatase
KLF
PI4K
CRISPR/Cas9
Aquaporin
SGK
Anti-infection
NOD
BMI-1
PKM

Keywords