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Clinical Compound Library

Catalog No. L3400
  Library Compound List   Excel SDF

Clinical compound library is a collection of 3142 compounds, all of which have been permitted into the clinical trial phases. These compounds have known biological activities, low toxicity, and clear mechanism with demonstrated pre-clinical evidence.

Every compound contains detailed information on pharmacological activities, targets, clinical development status, and indications with broad spectrum covering several therapeutic areas from cancer, inflammation, infection, neuropsychiatry to cardiology, and many drug targets such as JAK, EGFR, mTOR, CDK, HDAC, AKT, PARP, etc. It is an effective tool for drug screening as well as for cell differentiation induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
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Product Description

  • A unique collection of 3142 compounds in clinical trial phases for high throughput screening (HTS) and high content screening (HCS);
  • All compounds have been permitted into clinical trial phases, categorized into Phase 1, Phase 2 and Phase 3.
  • An effective tool for new drug screening and cell differentiation induction;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L3400)

Library Composition

Autophagy (385)
Apoptosis (353)
Antibacterial (243)
Antibiotic (236)
Endogenous Metabolite (220)
5-HT Receptor (138)
Adrenergic Receptor (110)
DNA/RNA Synthesis (93)
Dopamine Receptor (88)
HIV Protease (85)
AChR (82)
COX (78)
VEGFR (68)
Parasite (66)
Histamine Receptor (63)
Sodium Channel (61)
PI3K (60)
Antifungal (60)
Calcium Channel (59)
Potassium Channel (59)
EGFR (53)
P450 (49)
FLT (49)
Reactive Oxygen Species (47)
Topoisomerase (46)
Ferroptosis (46)
Glucocorticoid Receptor (45)
CDK (44)
PDE (44)
PDGFR (44)
SARS-CoV (43)
Dehydrogenase (43)
JAK (43)
Influenza Virus (41)
HDAC (41)
HCV Protease (41)
FGFR (40)
c-Kit (40)
Microtubule Associated (39)
Estrogen/progestogen Receptor (39)
PPAR (38)
GABA Receptor (37)
mTOR (37)
Mitophagy (35)
c-Met/HGFR (34)
RAAS (34)
Prostaglandin Receptor (32)
Src (32)
NF-κB (32)
Nucleoside Antimetabolite/Analog (30)
Reverse Transcriptase (30)
HBV (28)
Bcr-Abl (26)
Adenosine Receptor (26)
Proteasome (26)
Raf (24)
Androgen Receptor (23)
GPR (23)
Tyrosine Kinases (23)
Virus Protease (22)
Serotonin Transporter (22)
ROS (21)
Akt (20)
HSV (20)
iGluR (20)
Epigenetic Reader Domain (20)
HSP (19)
DNA Alkylator/Crosslinker (19)
Phosphatase (19)
PARP (19)
MEK (19)
Opioid Receptor (19)
BTK (19)
Estrogen Receptor/ERR (19)
ribosome (18)
Mitochondrial Metabolism (18)
NMDAR (18)
Norepinephrine (18)
Progesterone Receptor (18)
P-gp (17)
ALK (17)
TNF (17)
HER (17)
c-RET (17)
p38 MAPK (17)
Antifection (17)
Beta Amyloid (17)
Transferase (16)
IL Receptor (16)
Trk receptor (16)
Carbonic Anhydrase (15)
ATPase (15)
Retinoid Receptor (15)
Antioxidant (15)
AChE (15)
ERK (15)
Gamma-secretase (14)
Glucagon Receptor (14)
GluR (14)
PKC (14)
TAM Receptor (14)
Interleukin (14)
DPP-4 (14)
E1/E2/E3 Enzyme (14)
Aurora Kinase (14)
Thrombin (13)
GSK-3 (13)
HIF/HIF Prolyl-Hydroxylase (13)
CXCR (13)
BCL (13)
c-Fms (13)
TRP/TRPV Channel (13)
Proton pump (12)
Chk (12)
GNRH Receptor (12)
Antifolate (12)
DNA Alkylation (12)
Guanylate cyclase (12)
Caspase (12)
AMPK (12)
STAT (12)
NO Synthase (12)
DNA-PK (12)
Glucokinase (12)
Endothelin Receptor (12)
S1P Receptor (11)
CFTR (11)
MMP (11)
CCR (11)
MRP (11)
TLR (11)
Thyroid hormone receptor(THR) (11)
NADPH (10)
Syk (10)
P2 Receptor (10)
p53 (10)
MAO (10)
LPL Receptor (10)
FAK (10)
Phospholipase (10)
Integrin (10)
CSF-1R (10)
HMG-CoA Reductase (10)
Vasopressin Receptor (10)
HIF (10)
OX Receptor (9)
Lipoxygenase (9)
PLK (9)
Hedgehog/Smoothened (9)
S6 Kinase (9)
Sigma receptor (9)
Antiviral (9)
DNA Methyltransferase (9)
SGLT (9)
IGF-1R (9)
Cannabinoid Receptor (8)
DHFR (8)
DNA (8)
Glutathione Peroxidase (8)
Monoamine Oxidase (8)
Neurokinin receptor (8)
Sirtuin (8)
Wnt/beta-catenin (8)
PKA (8)
Histone Methyltransferase (8)
Hydroxylase (8)
IAP (8)
ROCK (8)
Xanthine Oxidase (7)
TGF-beta/Smad (7)
Drug Metabolite (7)
Mdm2 (7)
Serine Protease (7)
Reductase (7)
Aryl Hydrocarbon Receptor (7)
Ras (7)
Indoleamine 2,3-Dioxygenase (IDO) (7)
FXR (7)
ATM/ATR (7)
JNK (7)
RSV (6)
PAK (6)
Smo (6)
LTR (6)
Kinesin (6)
Beta-Secretase (6)
Aminopeptidase (6)
Complement System (6)
CAT (6)
IκB/IKK (6)
Isocitrate Dehydrogenase (IDH) (6)
Casein Kinase (6)
CETP (6)
NOS (6)
AhR (6)
Amino Acids and Derivatives (5)
RIP kinase (5)
Acyltransferase (5)
CaMK (5)
Pim (5)
BACE (5)
Ephrin Receptor (5)
Factor Xa (5)
Fatty Acid Synthase (5)
Gap Junction Protein (5)
IDO (5)
Leukotriene Receptor (5)
DNA gyrase (5)
Histone Demethylase (5)
ROR (4)
Decarboxylase (4)
Tie-2 (4)
Bradykinin Receptor (4)
GHSR (4)
DprE1 (4)
Liver X Receptor (4)
Chloride channel (4)
FAAH (4)
CaSR (4)
Melatonin Receptor (4)
CGRP Receptor (4)
Monoamine Transporter (4)
Neprilysin (4)
Somatostatin (4)
Aromatase (4)
IFNAR (4)
Oxytocin Receptor (4)
PGE Synthase (3)
PDK (3)
MT Receptor (3)
Serine/threonin kinase (3)
KSP (3)
Cysteine Protease (3)
IRAK (3)
ABC (3)
Rho (3)
Arginase (3)
GPCR19 (3)
Myosin (3)
Adenosine deaminase (3)
OAT (3)
NOD-like Receptor (NLR) (3)
Nrf2 (3)
STING (3)
cholecystokinin (3)
Tyrosinase (3)
Neuropeptide Y Receptor (3)
Free radical scavengers (3)
Telomerase (3)
NAMPT (3)
CRM1 (3)
Acetyl-CoA Carboxylase (3)
NADPH-oxidase (3)
VDA (2)
UGT (2)
Stearoyl-CoA Desaturase (SCD) (2)
Histone Acetyltransferase (2)
Anti-infection (2)
Hexokinase (2)
Discoidin Domain Receptor (DDR) (2)
DUB (2)
Galectin (2)
Annexin A (2)
GlyT (2)
GST (2)
Taste receptor (2)
YAP (2)
PAI-1 (2)
Porcupine (2)
c-Myc (2)
LPA Receptor (2)
MAPK (2)
NEDD8 (2)
LDL (2)
BCRP (2)
Na-K-Cl cotransporter (2)
CRFR (2)
IRE1 (2)
P2X Receptor (2)
ATP Citrate Lyase (2)
Melanocortin Receptor (2)
Protease-activated Receptor (2)
Integrase (2)
PYK2 (2)
Cell wall (2)
advanced glycation end products (1)
OXPHOS (1)
MELK (1)
Thioredoxin (1)
TOPK (1)
FLAP (1)
transporter (1)
NPC1L1 (1)
MLK (1)
NOD (1)
DYRK (1)
MNK (1)
VDAC (1)
ACK (1)
Wee1 (1)
Monocarboxylate transporter (1)
N-Acetylglucosaminyltransferase (1)
GluCls (1)
ASK (1)
p97 (1)
LHRH (1)
CRISPR/Cas9 (1)
Aquaporin (1)
Hydrogenase (1)
PKM (1)
KLF (1)
PI4K (1)
Hck (1)
BMI-1 (1)
PERK (1)
SGK (1)
GTPase (1)
Glutaminase (1)
Lipase (1)
GSNOR (1)
Anion Exchanger (1)
PD-1/PD-L1 (1)
GRK (1)
Lipid (1)
Stemness kinase (1)
RAR/RXR  (1)
Survivin (1)
PAFR (1)
Pyroptosis (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE