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Failed Clinical Trials Compound Library
Catalog No. L3420
TargetMol Clinical Failed Compounds Library compiles 1332 drug molecules from clinical trials marked as TERMINATED or WITHDRAWN in the ClinicalTrials database. Although these drugs did not achieve success in their original indications, they have undergone varying degrees of human studies, accumulating valuable data on safety and preliminary efficacy. Each compound is accompanied by detailed target information, activity descriptions, and indications. The drugs in the Failed Clinical Trials Compound Library possess good safety profiles and bioavailability, making them an important resource for repurposing old drugs. They can significantly increase the success rate of drug development, while shortening the development cycle and low-cost..
All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
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Contact us for more batch informationCatalog No. L3420
Failed Clinical Trials Compound LibrarysizeIn stock
- 1 mg
- 30 μL x 10 mM (in DMSO)
- 50 μL x 10 mM (in DMSO)
- 100 μL x 10 mM (in DMSO)
- 250 μL x 10 mM (in DMSO)
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Product Description
- A unique collection of 1332 clinical failed compounds for high throughput screening (HTS) and high content screening (HCS);
- Covers various research areas: oncology, cardiovascular drugs, nervous system drugs, respiratory system drugs, etc.
- More detailed compound information with structure, target, activity, IC50 value, and brief introduction;
- Structurally diverse, medicinally active, and cell permeable;
- NMR and HPLC validated to ensure high purity and quality;
Packaging And Storage
- Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
- Shipped with blue ice
Library Customization
Targetmol Compound Libraries
can be highly customized!
Inquiry & Customcan be highly customized!
Library Composition
Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Adrenergic Receptor
Dopamine Receptor
Endogenous Metabolite
HIV Protease
DNA/RNA Synthesis
Histamine Receptor
AChR
VEGFR
Parasite
FLT
Potassium Channel
Sodium Channel
c-Kit
PDGFR
EGFR
Calcium Channel
Antifungal
PI3K
COX
Dehydrogenase
JAK
SARS-CoV
Topoisomerase
Cytochromes P450
Influenza Virus
Microtubule Associated
Src
Ferroptosis
FGFR
Serotonin Transporter
PDE
c-Met/HGFR
RAAS
PPAR
Bcr-Abl
Epigenetic Reader Domain
mTOR
Mitophagy
Nucleoside Antimetabolite/Analog
CDK
HSP
Estrogen/progestogen Receptor
PKC
Glucocorticoid Receptor
Opioid Receptor
Reactive Oxygen Species
HDAC
Norepinephrine
NF-κB
HER
Proteasome
Phosphatase
HBV
Tyrosine Kinases
MAO
Endothelin Receptor
Aurora Kinase
Antiviral
Prostaglandin Receptor
Reverse Transcriptase
HCV Protease
PARP
Raf
NMDAR
Androgen Receptor
Akt
c-Fms
ribosome
GABA Receptor
Progesterone Receptor
iGluR
Vasopressin Receptor
GPR
c-RET
Neurokinin receptor
TAM Receptor
Thrombin
Proton pump
HSV
Trk receptor
Nrf2
ALK
Beta Amyloid
Retinoid Receptor
Phospholipase
TNF
Monoamine Oxidase
ATPase
Adenosine Receptor
Virus Protease
CSF-1R
IAP
Gamma-secretase
ROS
CXCR
Indoleamine 2,3-Dioxygenase (IDO)
P-gp
Hydroxylase
HMG-CoA Reductase
S1P Receptor
Carbonic Anhydrase
DHFR
Antioxidant
LPL Receptor
DNA Alkylator/Crosslinker
Factor Xa
Estrogen Receptor/ERR
Serine Protease
Antifolate
FXR
Caspase
TRP/TRPV Channel
ERK
ROCK
E1/E2/E3 Enzyme
Guanylate cyclase
DPP-4
Hedgehog/Smoothened
CCR
MMP
GluR
TLR
Ephrin Receptor
Bcl-2 Family
STAT
PLK
MEK
Cannabinoid Receptor
Syk
ADC Cytotoxin
P2Y Receptor
BACE
Histone Demethylase
GNRH Receptor
MRP
P2X Receptor
Mitochondrial Metabolism
Antifection
Molecular Glues
Smo
DNA Alkylation
IL Receptor
IGF-1R
CaMK
Interleukin
SGLT
Beta-Secretase
Ligand for E3 Ligase
HIF
DNA Methyltransferase
S6 Kinase
HIF/HIF Prolyl-Hydroxylase
ROS Kinase
Thyroid hormone receptor(THR)
Transferase
Histone Methyltransferase
Integrin
CETP
GSK-3
Kisspeptin
Glucokinase
Aryl Hydrocarbon Receptor
IDO
RIP kinase
GlyT
PAK
OX Receptor
DNA
Aminopeptidase
transporter
Decarboxylase
RSV
ATM/ATR
GST
AMPK
Oxytocin Receptor
GHSR
NADPH-oxidase
AhR
Imidazoline Receptor
p53
PD-1/PD-L1
NO Synthase
BTK
Mdm2
NOS
ROR
NEDD8
CRM1
p38 MAPK
Ligands for Target Protein for PROTAC
Reductase
IFNAR
Glutathione Peroxidase
Melatonin Receptor
c-Myc
CaSR
PKA
Pim
Rho
Serine/threonin kinase
Leukotriene Receptor
Myosin
IRE1
Drug Metabolite
MT Receptor
DNA gyrase
ABC Transporter
Integrase
Fatty Acid Synthase
Thrombopoietin Receptor
Lipoxygenase
TGF-beta/Smad
Wee1
Acyltransferase
GPCR19
GluCls
CRFR
Casein Kinase
IκB/IKK
Aromatase
Adenosine Deaminase
IRAK
Ras
Sigma receptor
p97
FAK
NOD-like Receptor (NLR)
Advanced Glycation End Products
NPC1L1
DNA-PK
Amino Acids and Derivatives
DprE1
YAP
Cell wall
NADPH
Lipase
JNK
gp120/CD4
Tie-2
VDA
Cholecystokinin Receptor
Wnt/beta-catenin
Hck
Cysteine Protease
Liver X Receptor
NAMPT
Glutaminase
SIK
FLAP
PAFR
LDL
Glucagon Receptor
Na-K-Cl cotransporter
Hexokinase
Monoamine Transporter
Isocitrate Dehydrogenase (IDH)
Thioredoxin
FAAH
Bradykinin Receptor
Cholinesterase (ChE)
Somatostatin
Chk
Xanthine Oxidase
KSP
DUB
ATP Citrate Lyase
PGE Synthase
MAPK
MNK
STING
Sirtuin
Histone Acetyltransferase
PAI-1
Pyroptosis
Methionine Adenosyltransferase (MAT)
Hippo pathway
Acetyl-CoA Carboxylase
GPX
LPA Receptor
KLF
PI4K
PDK
Aquaporin
Complement System
Discoidin Domain Receptor (DDR)
Gap Junction Protein
NOD
Tyrosinase
Protease-activated Receptor
MLK
Kinesin
Vitamin
Library Information
| Empty | 99755-59-6 | 99009-20-8 | 98-96-4 | 987-78-0 | 98769-84-7 | 98717-15-8 | 985-12-6 | 98319-26-7 | 980-71-2 | 97-77-8 | Empty |
| Rotigotine- | Pyrazoloacridine | Pyrazinamide | Citicoline | Reboxetine mesylate | Ropivacaine hydrochloride | Drotaverine hydrochloride | Finasteride | Brompheniramine maleate | Disulfiram | ||
| Empty | 97657-92-6 | 96187-53-0 | 960404-48-2 | 96036-03-2 | 96020-91-6 | 960203-27-4 | 958852-01-2 | 95809-78-2 | 957054-30-7 | 956905-27-4 | Empty |
| Latrepirdine dihydrochloride | Brequinar | Dapagliflozin ((2S)-1,2-propanediol, hydrate) | Meropenem | Eflornithine hydrochloride hydrate | Vortioxetine hydrobromide | GSK1059615 | Devimistat | Pictilisib | PF-04217903 | ||
| Empty | 956483-03-7 | 95635-56-6 | 95635-55-5 | 956104-40-8 | 955365-80-7 | 954126-98-8 | 953769-46-5 | 953428-73-4 | 950769-58-1 | 95058-81-4 | Empty |
| FV-100 | Ranolazine dihydrochloride | Ranolazine | Apalutamide | Adavosertib | Danirixin | Sotuletinib | JNJ-39393406 | Quizartinib | Gemcitabine | ||
| Empty | 947331-05-7 | 945755-56-6 | 945635-15-4 | 945531-77-1 | 94497-51-5 | 944396-07-0 | 943540-75-8 | 943319-70-8 | 942123-43-5 | 94-16-6 | Empty |
| Allisartan Isoproxil | XL019 | Deferitazole | Ezutromid | Tamibarotene | Buparlisib | JNJ-38877605 | Ponatinib | Inarigivir soproxil | Aminohippurate sodium | ||
| Empty | 93957-55-2 | 937272-79-2 | 937174-76-0 | 936563-96-1 | 936539-80-9 | 936500-94-6 | 936091-26-8 | 935888-69-0 | 935881-37-1 | 935840-31-6 | Empty |
| Fluvastatin sodium | Pacritinib | GSK-690693 | Ibrutinib | Betrixaban maleate | Elinogrel | Fedratinib | Oprozomib | AR42 | PF-03654746 | ||
| Empty | 935666-88-9 | 935283-04-8 | 93265-81-7 | 929016-96-6 | 928659-17-0 | 92823-03-5 | 928037-13-2 | 926927-61-9 | 92-62-6 | 925206-65-1 | Empty |
| AZD-1480 | Linzagolix | Ropidoxuridine | Pracinostat | Triazavirin | Flomoxef sodium | Golvatinib | Motolimod | Proflavine | RRX-001 | ||
| Empty | 923564-51-6 | 923359-38-0 | 923288-95-3 | 923288-90-8 | 923262-96-8 | 923032-37-5 | 920113-03-7 | 918639-08-4 | 918407-35-9 | 916151-99-0 | Empty |
| Navitoclax | SAR407899 | Nilotinib hydrochloride | Nilotinib monohydrochloride monohydrate | SAR407899 hydrochloride | Refametinib | Riviciclib hydrochloride | Bosutinib hydrate | Avoralstat | APTO-253 | ||
| Empty | 915942-22-2 | 915769-50-5 | 915385-81-8 | 915020-55-2 | 915019-65-7 | 914453-95-5 | 91374-20-8 | 912999-49-6 | 911714-45-9 | 91161-71-6 | Empty |
| Neratinib maleate | Dovitinib lactate hydrate | Opaganib | BGT226 | Dactolisib | Atosiban acetate | Ropinirole hydrochloride | Onalespib | SP-420 | Terbinafine |
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