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FDA-Approved Drug Library

Catalog No. L4200
  Library Compound List   Excel SDF

All compounds in FDA approved drug library have well-characterized biological activity, clear targets, safety, and bioavailability – properties which could dramatically accelerate drug development and optimization. It is an effective and ideal tool for drug repurposing and cell differentiation induction. Detailed information on each compound in this library can help scientists quickly finish drug screening or make quick judgement on cell differentiation mechanism, and create conditions for further investigation on the mechanism of action.

In addtion, we put the compounds that should be provided in the form of dry powder together to form Part B in order to ensure the best using effect of the compound library and increase the probability of successful screening as much as possible.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Please contact us for prices and availability for the specification of product you are interested at.
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If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 1729 FDA approved drugs for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety confirmed by pre-clinical research evidence and clinical trials;
  • An effective tool for discovering new with old drugs and new drug target identification;
  • Covers various research areas: oncology, cardiology, anti-inflammatory, immunology, neuropsychiatry, analgesia etc
  • Structurally diverse, medicinally active, and cell permeable;
  • Rich documentation with structure, target, IC50 value and biological activity description;
  • NMR and HPLC/LCMS validated to ensure high purity.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L4200)

Library Composition

Antibacterial (260)
Antibiotic (257)
Autophagy (248)
Apoptosis (162)
Endogenous Metabolite (129)
Adrenergic Receptor (120)
5-HT Receptor (111)
AChR (91)
Dopamine Receptor (73)
Histamine Receptor (66)
HIV Protease (64)
DNA/RNA Synthesis (59)
Sodium Channel (57)
COX (54)
Antifungal (51)
Parasite (50)
Potassium Channel (47)
Glucocorticoid Receptor (43)
Calcium Channel (38)
Estrogen/progestogen Receptor (37)
P450 (34)
Topoisomerase (33)
Ferroptosis (33)
RAAS (27)
ribosome (26)
SARS-CoV (25)
GABA Receptor (25)
Serotonin Transporter (25)
Dehydrogenase (24)
VEGFR (24)
PDE (24)
Mitophagy (23)
c-Kit (23)
Nucleoside Antimetabolite/Analog (22)
Microtubule Associated (22)
Reverse Transcriptase (22)
HCV Protease (22)
Antifection (21)
Norepinephrine (20)
PDGFR (20)
Progesterone Receptor (18)
Influenza Virus (18)
Reactive Oxygen Species (18)
EGFR (18)
HSV (18)
DNA Alkylator/Crosslinker (17)
PPAR (16)
Estrogen Receptor/ERR (16)
Androgen Receptor (15)
Proton pump (15)
AChE (14)
Carbonic Anhydrase (14)
Prostaglandin Receptor (14)
Proteasome (14)
Opioid Receptor (13)
FLT (13)
HBV (13)
MAO (13)
ATPase (13)
GNRH Receptor (12)
Thrombin (12)
Adenosine Receptor (12)
FGFR (11)
c-Met/HGFR (11)
Monoamine Oxidase (11)
Raf (11)
MRP (11)
ROS (11)
HDAC (11)
Virus Protease (11)
DHFR (10)
TRP/TRPV Channel (10)
c-RET (10)
Antifolate (10)
iGluR (10)
Src (10)
JAK (10)
Phosphatase (9)
ALK (9)
HMG-CoA Reductase (9)
Bcr-Abl (9)
Drug Metabolite (9)
Tyrosine Kinases (9)
NF-κB (9)
Thyroid hormone receptor(THR) (8)
Retinoid Receptor (8)
Phospholipase (8)
NO Synthase (8)
CaMK (8)
Transferase (8)
P2 Receptor (8)
GluR (8)
Guanylate cyclase (7)
CDK (7)
P-gp (7)
DPP-4 (7)
ABC (7)
MMP (7)
NMDAR (7)
DNA Alkylation (7)
DNA gyrase (7)
Factor Xa (7)
PI3K (7)
HER (6)
PARP (6)
PKC (6)
STAT (6)
TNF (6)
Glucagon Receptor (6)
MEK (6)
Lipoxygenase (6)
mTOR (6)
Neurokinin receptor (5)
NADPH (5)
Monoamine Transporter (5)
SGLT (5)
TAM Receptor (5)
LPL Receptor (5)
S1P Receptor (5)
Histone Methyltransferase (5)
CFTR (5)
Hedgehog/Smoothened (5)
DNA (5)
GPR (5)
DNA Methyltransferase (5)
Trk receptor (5)
Cell wall (5)
CAT (5)
Endothelin Receptor (5)
Reductase (4)
Ras (4)
Histone Demethylase (4)
ADC Cytotoxin (4)
CaSR (4)
AMPK (4)
Glutathione Peroxidase (4)
Antiviral (4)
TLR (4)
IL Receptor (4)
Aromatase (4)
Neprilysin (3)
BTK (3)
Vasopressin Receptor (3)
Somatostatin (3)
BCL (3)
Sigma receptor (3)
AhR (3)
Smo (3)
MT Receptor (3)
Chloride channel (3)
GST (3)
Complement System (3)
FXR (3)
Serine Protease (3)
Hydroxylase (3)
ROCK (3)
IGF-1R (3)
Integrin (3)
Amino Acids and Derivatives (3)
Fatty Acid Synthase (3)
ERK (3)
Leukotriene Receptor (3)
PAK (3)
Decarboxylase (3)
Cysteine Protease (3)
Mitochondrial Metabolism (3)
RSV (2)
Xanthine Oxidase (2)
Rho (2)
Protease-activated Receptor (2)
Oxytocin Receptor (2)
Adenosine deaminase (2)
Aryl Hydrocarbon Receptor (2)
Wnt/beta-catenin (2)
Tyrosinase (2)
Gamma-secretase (2)
Free radical scavengers (2)
Ephrin Receptor (2)
Annexin A (2)
CXCR (2)
CRM1 (2)
cholecystokinin (2)
NOS (2)
CGRP Receptor (2)
c-Fms (2)
UGT (2)
CCR (2)
Caspase (2)
Arginase (2)
Beta Amyloid (2)
Gap Junction Protein (2)
Glutathione reductase (2)
GPCR19 (2)
GSK-3 (2)
Syk (2)
Melatonin Receptor (2)
Melanocortin Receptor (2)
LTR (2)
Lipid (2)
LDL (2)
Isocitrate Dehydrogenase (IDH) (2)
IRE1 (2)
Interleukin (2)
Integrase (2)
HSP (2)
HIF/HIF Prolyl-Hydroxylase (2)
Thrombopoietin Receptor (2)
Telomerase (1)
TGF-beta/Smad (1)
VDA (1)
Sirtuin (1)
IAP (1)
ROR (1)
CRISPR/Cas9 (1)
GlyT (1)
Glucokinase (1)
FAAH (1)
Epigenetic Reader Domain (1)
DUB (1)
CSF-1R (1)
Chk (1)
HIF (1)
CETP (1)
Bradykinin Receptor (1)
Beta-Secretase (1)
ATP Citrate Lyase (1)
Angiotensin-converting Enzyme (ACE) (1)
Akt (1)
ACK (1)
GRK (1)
Histone Acetyltransferase (1)
RAR/RXR  (1)
OAT (1)
Pyroptosis (1)
PLK (1)
PKM (1)
Phosphorylase (1)
PGE Synthase (1)
PDK (1)
OX Receptor (1)
Nrf2 (1)
Hydrogenase (1)
NPC1L1 (1)
NOD-like Receptor (NLR) (1)
Na-K-Cl cotransporter (1)
NADPH-oxidase (1)
MTH1 (1)
MAPK (1)
IκB/IKK (1)
YAP (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE