Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Kinase Inhibitor Library

Catalog No. L1600

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. A protein kinase modifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved in signal transduction. Various other kinases act on small molecules such as lipids, carbohydrates, amino acids, and nucleotides, either for signaling or to prime them for metabolic pathways. TargetMol’s Kinase Inhibitor Library, containing 2840 kinase inhibitors/regulators , can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L1600

Kinase Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Product Description Product Description

  • A unique collection of 2840 kinase inhibitors for high throughput screening and high content screening for drug discovery in kinase related diseases;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include MAPK, PI3K, JAK, STAT, CDK, MEK, Insulin/IGF receptors, CaM Kinease II, PKA, JNK, PKC, RAF, EGFR, SAPK, GSK, MLCK, Src-family, IKK, PDGFR, VEGFR, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Library Customization | TargetMol Library Composition

Apoptosis
CDK
Autophagy
EGFR
PI3K
VEGFR
mTOR
JAK
FLT
Src
PDGFR
GSK-3
Raf
FGFR
c-Kit
PKC
Bcr-Abl
c-Met/HGFR
Akt
p38 MAPK
ALK
ERK
BTK
Aurora Kinase
ROCK
Kras
AMPK
Ras
Tyrosine Kinases
MAPK
PKA
Casein Kinase
MEK
DNA-PK
Serine/threonin kinase
c-RET
IGF-1R
TAM Receptor
RIP kinase
CaMK
Trk receptor
Epigenetic Reader Domain
IκB/IKK
FAK
Glucokinase
JNK
TGF-beta/Smad
S6 Kinase
ATM/ATR
c-Fms
PLK
HER
Chk
PERK
Syk
Pim
LRRK2
IRAK
ROR
DYRK
Rho
PDK
Wnt/beta-catenin
PAK
PI4K
NF-κB
PROTACs
IRE1
Ephrin Receptor
Mitophagy
Parasite
STAT
ROS Kinase
Calcium Channel
Phosphatase
Glucosidase
Antibacterial
Tyrosinase
Ferroptosis
CSF-1R
GRK
Influenza Virus
TNF
Discoidin Domain Receptor (DDR)
MNK
Microtubule Associated
MLK
HIV Protease
Serine Protease
LIM Kinase
Adrenergic Receptor
SGK
Potassium Channel
AChR
Kinesin
PDE
ROS
DNA/RNA Synthesis
Endogenous Metabolite
5-HT Receptor
S1P Receptor
Dehydrogenase
Tie-2
PYK2
SIK
AAK1 (AP2 associated kinase 1)
Interleukin
Wee1
Antiviral
Antibiotic
PKM
Histone Methyltransferase
Adenosine Receptor
Virus Protease
PPAR
Drug Metabolite
Mitochondrial Metabolism
BCL
COX
SARS-CoV
MELK
HDAC
DAPK
Sodium Channel
Dopamine Receptor
HCV Protease
Histamine Receptor
TOPK
Caspase
TRP/TRPV Channel
IL Receptor
ACK
ASK
Hippo pathway
P450
Integrin
Ligands for Target Protein for PROTAC
GTPase
Myosin
DNA Alkylation
HSV
Carboxypeptidase
Beta Amyloid
Carbonic Anhydrase
Transferase
YAP
Antifungal
LPL Receptor
IFNAR
Hck
Topoisomerase
E1/E2/E3 Enzyme
Haspin Kinase
Hexokinase
Reactive Oxygen Species
P-gp
cholecystokinin
Antioxidant
BACE
Histone Demethylase
Estrogen Receptor/ERR
PARP
Serotonin Transporter
Aryl Hydrocarbon Receptor
MMP
cAMP
GluR
DUB
HSP
transporter
Nrf2
PAI-1
Reverse Transcriptase
CRISPR/Cas9
GPR
Phospholipase
Cannabinoid Receptor
NO Synthase
Apelin receptor
ATPase
Chloride channel
Proton pump
NOS
DHFR
MyD88
Estrogen/progestogen Receptor
RAR/RXR 
NADPH
RAAS
Necroptosis
Glutathione Peroxidase
HBV
Antifolate
Nucleoside Antimetabolite/Analog
Liver X Receptor
FXR
NAMPT
Stemness kinase
MAO
Immunology/Inflammation related
iGluR
Gamma-secretase
LDL
Phosphorylase
P2X Receptor
NMDAR
Monoamine Transporter
Molecular Glues
Opioid Receptor
Fatty Acid Synthase
Thrombopoietin Receptor
Lipoxygenase
Norepinephrine
DNA
Indoleamine 2,3-Dioxygenase (IDO)
ATP Citrate Lyase
Lipid
BCRP
Beta-Secretase
Acyltransferase
Porcupine
STING
TLR
Sirtuin
Histone Acetyltransferase
Decarboxylase
cGAS
RSV
GPX
Retinoid Receptor
Ligand for E3 Ligase
Protease
Hydroxylase
HIF
RXFP receptor
Fer/FerT kinase
Gap Junction Protein
Anti-infection
NADPH-oxidase
BMI-1
Sigma receptor
Protease-activated Receptor
p97
HIF/HIF Prolyl-Hydroxylase
p53
PD-1/PD-L1