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TargetMol | Compound Library

Kinase Inhibitor Library

Catalog No. L1600

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. A protein kinase modifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved in signal transduction. Various other kinases act on small molecules such as lipids, carbohydrates, amino acids, and nucleotides, either for signaling or to prime them for metabolic pathways. TargetMol’s Kinase Inhibitor Library, containing 2900 kinase inhibitors/regulators , can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L1600

Kinase Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 2900 kinase inhibitors for high throughput screening and high content screening for drug discovery in kinase related diseases;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include MAPK, PI3K, JAK, STAT, CDK, MEK, Insulin/IGF receptors, CaM Kinease II, PKA, JNK, PKC, RAF, EGFR, SAPK, GSK, MLCK, Src-family, IKK, PDGFR, VEGFR, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
CDK
PI3K
EGFR
VEGFR
mTOR
JAK
Akt
p38 MAPK
Src
ERK
FLT
PKC
PDGFR
AMPK
GSK-3
FGFR
Raf
c-Kit
NF-κB
c-Met/HGFR
Bcr-Abl
ALK
BTK
MAPK
JNK
Aurora Kinase
Ras
PKA
Kras
Tyrosine Kinases
ROCK
MEK
Casein Kinase
Serine/threonin kinase
IGF-1R
Antibacterial
Endogenous Metabolite
Glucosidase
CaMK
c-RET
FAK
DNA-PK
RIP kinase
TAM Receptor
Trk receptor
IκB/IKK
S6 Kinase
TGF-beta/Smad
STAT
PLK
PERK
Glucokinase
ATM/ATR
c-Fms
TNF
Syk
HER
Parasite
Chk
Pim
IRAK
ROR
DYRK
Caspase
COX
LRRK2
Wnt/beta-catenin
PDK
Antibiotic
Mitophagy
HIV Protease
PAK
Influenza Virus
Rho
Ephrin Receptor
Tyrosinase
ROS Kinase
Phosphatase
Calcium Channel
IRE1
Reactive Oxygen Species
IL Receptor
Bcl-2 Family
PI4K
PROTACs
DNA/RNA Synthesis
Ferroptosis
PPAR
MMP
AChR
ROS
Epigenetic Reader Domain
S1P Receptor
Dehydrogenase
Antifungal
Adrenergic Receptor
CSF-1R
PDE
GRK
Cytochromes P450
MNK
Antiviral
5-HT Receptor
Potassium Channel
Discoidin Domain Receptor (DDR)
Kinesin
Beta Amyloid
Microtubule Associated
MLK
Adenosine Receptor
Serine Protease
LIM Kinase
HSV
HDAC
SGK
NO Synthase
Tie-2
PARP
SIK
Wee1
SARS-CoV
Nrf2
Sodium Channel
PKM
HCV Protease
Antioxidant
Virus Protease
AAK1
PYK2
Mitochondrial Metabolism
Cholinesterase (ChE)
Lipoxygenase
Interleukin
Histone Methyltransferase
Histamine Receptor
Topoisomerase
Drug Metabolite
Antifection
P-gp
MELK
DAPK
Dopamine Receptor
Integrin
LPL Receptor
TOPK
LDL
ACK1
TLR
transporter
ASK
Hippo pathway
Carbonic Anhydrase
Estrogen/progestogen Receptor
GTPase
Hck
TRP/TRPV Channel
Myosin
Hexokinase
DNA Alkylation
Carboxypeptidase
p53
ATPase
NOS
Transferase
Ligands for Target Protein for PROTAC
YAP
BACE
IFNAR
NADPH
Glutathione Peroxidase
HBV
Estrogen Receptor/ERR
Cholecystokinin Receptor
MAO
E1/E2/E3 Enzyme
Haspin Kinase
GluR
Indoleamine 2,3-Dioxygenase (IDO)
HSP
Prostaglandin Receptor
Sirtuin
PAI-1
GPR
Phospholipase
Cannabinoid Receptor
HIF/HIF Prolyl-Hydroxylase
Chloride channel
ADC Cytotoxin
Histone Demethylase
RAAS
gp120/CD4
Serotonin Transporter
Nucleoside Antimetabolite/Analog
FXR
Amylase
Aryl Hydrocarbon Receptor
Gamma-secretase
Monoamine Transporter
PTEN
cAMP
DUB
BCRP
Beta-Secretase
Reverse Transcriptase
CRISPR/Cas9
HIF
Anti-infection
NADPH-oxidase
Proteasome
Apelin receptor
Proton pump
NPC1L1
DHFR
MyD88
RAR/RXR 
Necroptosis
Melatonin Receptor
MRP
Antifolate
Cell Cycle Arrest
Liver X Receptor
NAMPT
Stemness kinase
Immunology/Inflammation related
iGluR
P2X Receptor
NMDAR
Molecular Glues
Opioid Receptor
Fatty Acid Synthase
Bombesin Receptor
Hedgehog/Smoothened
FAAH
PAD
Thrombopoietin Receptor
Norepinephrine
DNA
ATP Citrate Lyase
Lipid
PGE Synthase
Acyltransferase
Porcupine
STING
Histone Acetyltransferase
Decarboxylase
cGAS
RSV
GPX
Retinoid Receptor
Ligand for E3 Ligase
Protease
Aromatase
GABA Receptor
Hydroxylase
RXFP receptor
Gap Junction Protein
Fer/FerT kinase
BMI-1
NOD
Sigma receptor
Protease-activated Receptor
p97
PD-1/PD-L1