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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
Antibacterial
Antibiotic
5-HT Receptor
Adrenergic Receptor
Histamine Receptor
Dopamine Receptor
COX
AChR
HIV Protease
VEGFR
EGFR
DNA/RNA Synthesis
Potassium Channel
Parasite
Sodium Channel
Calcium Channel
PDE
PDGFR
P450
CDK
SARS-CoV
FLT
c-Kit
Estrogen/progestogen Receptor
Glucocorticoid Receptor
RAAS
Dehydrogenase
HCV Protease
PI3K
JAK
Src
Estrogen Receptor/ERR
FGFR
BTK
Antifungal
c-Met/HGFR
Bcr-Abl
PPAR
Serotonin Transporter
Ferroptosis
Reverse Transcriptase
HDAC
Proteasome
p38 MAPK
HBV
Topoisomerase
Androgen Receptor
Histone Methyltransferase
Epigenetic Reader Domain
Endogenous Metabolite
GPR
Microtubule Associated
Raf
GluR
Norepinephrine
Prostaglandin Receptor
ALK
GABA Receptor
TRP/TRPV Channel
Influenza Virus
HER
Phosphatase
Mitophagy
Tyrosine Kinases
PARP
NF-κB
Progesterone Receptor
iGluR
mTOR
Transferase
Adenosine Receptor
Opioid Receptor
Integrin
ERK
ROS
DPP-4
MAPK
MEK
Proton pump
Nucleoside Antimetabolite/Analog
Trk receptor
TNF
LPL Receptor
Factor Xa
GSK-3
Reactive Oxygen Species
MMP
Akt
P-gp
Antiviral
Kras
c-Fms
c-RET
Syk
TAM Receptor
Thrombin
S1P Receptor
Monoamine Oxidase
ROCK
NMDAR
Endothelin Receptor
SGLT
Retinoid Receptor
STAT
Carbonic Anhydrase
Reductase
HSV
CCR
CXCR
AChE
HSP
Beta Amyloid
HIF/HIF Prolyl-Hydroxylase
ATPase
MAO
Aurora Kinase
Lipoxygenase
Interleukin
Acyltransferase
ribosome
AMPK
Cannabinoid Receptor
ROS Kinase
Thyroid hormone receptor(THR)
DHFR
ADC Cytotoxin
MRP
Wnt/beta-catenin
PKC
CSF-1R
Gamma-secretase
Mitochondrial Metabolism
IL Receptor
ATM/ATR
Phospholipase
Virus Protease
Glucagon Receptor
Guanylate cyclase
Fatty Acid Synthase
IGF-1R
TGF-beta/Smad
Neurokinin receptor
ROR
NADPH
Histone Demethylase
E1/E2/E3 Enzyme
P2X Receptor
DNA gyrase
Hedgehog/Smoothened
RSV
Ligand for E3 Ligase
FAK
CFTR
DNA Alkylator/Crosslinker
P2Y Receptor
PKA
Antifolate
Serine/threonin kinase
Leukotriene Receptor
Caspase
Vasopressin Receptor
OX Receptor
Xanthine Oxidase
Beta-Secretase
TLR
Aromatase
Hydroxylase
PLK
Complement System
IRAK
HMG-CoA Reductase
Sigma receptor
NO Synthase
Mdm2
LTR
BACE
PERK
Glutathione Peroxidase
ABC
GNRH Receptor
Pim
Cysteine Protease
FXR
Antifection
Smo
BCL
DNA Alkylation
CaMK
transporter
ASK
Casein Kinase
GHSR
DNA Methyltransferase
Ras
PD-1/PD-L1
DNA-PK
Serine Protease
Isocitrate Dehydrogenase (IDH)
Stearoyl-CoA Desaturase (SCD)
Chk
Aminopeptidase
Ephrin Receptor
HIF
NADPH-oxidase
NOS
YAP
Lipase
Melatonin Receptor
IAP
Neuropeptide Y Receptor
PAK
FAAH
DNA
DUB
Indoleamine 2,3-Dioxygenase (IDO)
PGE Synthase
Porcupine
PAI-1
Neprilysin
cholecystokinin
Protease-activated Receptor
AhR
p53
Monocarboxylate transporter
CRM1
Antioxidant
IFNAR
CETP
JNK
TOPK
CaSR
Liver X Receptor
Glucokinase
Annexin A
FLAP
RIP kinase
Drug Metabolite
MT Receptor
Monoamine Transporter
Molecular Glues
PAD
Epoxide Hydrolase
Thrombopoietin Receptor
Mucin
OXPHOS
Free radical scavengers
IκB/IKK
GST
LPA Receptor
PI4K
Discoidin Domain Receptor (DDR)
NOD
S6 Kinase
Melanin-concentrating Hormone Receptor (MCHR)
advanced glycation end products
PROTACs
MALT
NEDD8
Ligands for Target Protein for PROTAC
Tie-2
Rho
Hck
Vitamin
Glutaminase
Aryl Hydrocarbon Receptor
IDO
SIK
IRE1
PAFR
GlyT
Hexokinase
Integrase
Bradykinin Receptor
Telomerase
Lipid
MNK
OAT
STING
LRRK2
Nrf2
Hippo pathway
Acetyl-CoA Carboxylase
PDK
Adenosine deaminase
CGRP Receptor
SGK
BMI-1
NOD-like Receptor (NLR)
MLK
Imidazoline Receptor
Kinesin
Chloride channel
Taste receptor
CAT
GSNOR
NPC1L1
CD38
Amino Acids and Derivatives
Na+/Ca2+ Exchanger
DYRK
Cell wall
Necroptosis
GTPase
c-Myc
Galectin
Neurotensin Receptor
NAMPT
PYK2
FOXO1
Prolyl Endopeptidase (PREP)
Myosin
Adiponectin receptor
UGT
Haspin Kinase
LDL
GRK
PACAP
AAK1 (AP2 associated kinase 1)
Na-K-Cl cotransporter
Glucosidase
PROTAC Linker
HCN Channel
Angiotensin-converting Enzyme (ACE)
Somatostatin
ACK
cAMP
ATP Citrate Lyase
Wee1
BCRP
Survivin
GPCR19
Sirtuin
Histone Acetyltransferase
Pyroptosis
Methionine Adenosyltransferase (MAT)
GPX
Melanocortin Receptor
CRISPR/Cas9
Oxytocin Receptor
RXFP receptor
Gap Junction Protein
Platelet aggregation
Anti-infection
Tyrosinase
p97
PKM

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