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TargetMol | Compound Library

Orally Active Compound Library

Catalog No. L9850

Oral administration is the first choice for clinical drug delivery, especially for long-term use. It is also the safest, most convenient, and most economical method of drug delivery. Oral bioavailability is the percentage of the absorbed drug dose successfully passed through the mucosa of the gastrointestinal tract and entered the bloodstream through the liver, to the original given oral dose. Drugs with high oral bioavailability can achieve efficacy at lower doses and effectively reduce toxic side effects; while when bioavailability is too low, even compounds with good pharmacological activity are unable to be fully exposed and utilized at the target site, resulting in therapeutic failure or high dose with large toxic side effects, which eventually leads to drug development failure and limits the application. TargetMol has carefully collected 3160 compounds with publicly reported oral activity that can be used for drug repurposing and development of orally active drugs.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L9850

Orally Active Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A unique collection of 3160 of orally active compounds for high-throughput screening and high-content screening.
  • Some drugs are approved or are in clinical trials with validated biological activity and safety.
  • Detailed specifications, compound structures, target information, activity descriptions, etc.
  • NMR and HPLC detection techniques to ensure high product purity.
  • All compounds are available in stock.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Autophagy
Apoptosis
Antibacterial
Antibiotic
5-HT Receptor
Endogenous Metabolite
Adrenergic Receptor
Histamine Receptor
Dopamine Receptor
COX
AChR
HIV Protease
Parasite
VEGFR
DNA/RNA Synthesis
Potassium Channel
EGFR
Sodium Channel
PDE
Calcium Channel
SARS-CoV
Estrogen/progestogen Receptor
Cytochromes P450
CDK
PDGFR
Glucocorticoid Receptor
Dehydrogenase
FLT
RAAS
c-Kit
PI3K
Antifungal
Estrogen Receptor/ERR
HCV Protease
Topoisomerase
JAK
Src
FGFR
Ferroptosis
Reactive Oxygen Species
Microtubule Associated
PPAR
BTK
Mitophagy
c-Met/HGFR
HBV
Bcr-Abl
Reverse Transcriptase
NF-κB
p38 MAPK
Serotonin Transporter
GluR
GABA Receptor
TRP/TRPV Channel
Androgen Receptor
Prostaglandin Receptor
Influenza Virus
Proteasome
iGluR
Epigenetic Reader Domain
HDAC
GPR
Histone Methyltransferase
Norepinephrine
Phosphatase
Tyrosine Kinases
Raf
ALK
Adenosine Receptor
Cholinesterase (ChE)
mTOR
Progesterone Receptor
HER
PARP
ROS
Transferase
Integrin
Opioid Receptor
HSV
MMP
MAPK
Antiviral
ribosome
TNF
GSK-3
ERK
DPP-4
Kras
Thrombin
HIF/HIF Prolyl-Hydroxylase
S1P Receptor
Proton pump
LPL Receptor
Factor Xa
Nucleoside Antimetabolite/Analog
NMDAR
P-gp
Trk receptor
Beta Amyloid
Virus Protease
Retinoid Receptor
STAT
c-Fms
MEK
c-RET
Syk
Monoamine Oxidase
ROCK
MAO
Mitochondrial Metabolism
Endothelin Receptor
Aurora Kinase
Lipoxygenase
SGLT
Akt
Carbonic Anhydrase
ADC Cytotoxin
Reductase
MRP
CCR
CXCR
HSP
Phospholipase
Cannabinoid Receptor
TAM Receptor
Thyroid hormone receptor(THR)
ATPase
Wnt/beta-catenin
Gamma-secretase
DNA gyrase
Fatty Acid Synthase
IL Receptor
Interleukin
Acyltransferase
ROS Kinase
DHFR
NADPH
PKC
CSF-1R
ATM/ATR
AMPK
ROR
Caspase
Glucagon Receptor
P2X Receptor
Guanylate cyclase
IGF-1R
TGF-beta/Smad
TLR
Neurokinin receptor
HMG-CoA Reductase
CFTR
NO Synthase
Antioxidant
Histone Demethylase
Glutathione Peroxidase
PKA
E1/E2/E3 Enzyme
ABC Transporter
Antifection
Hedgehog/Smoothened
Bcl-2 Family
RSV
PLK
Complement System
FAK
P2Y Receptor
LTR
Serine/threonin kinase
Cysteine Protease
FXR
Leukotriene Receptor
Vasopressin Receptor
OX Receptor
Xanthine Oxidase
CaMK
Beta-Secretase
Aminopeptidase
Nrf2
Ligand for E3 Ligase
Aromatase
Hydroxylase
HIF
IRAK
Sigma receptor
Mdm2
DNA Alkylator/Crosslinker
BACE
PERK
GNRH Receptor
Pim
Antifolate
IAP
Smo
Indoleamine 2,3-Dioxygenase (IDO)
transporter
ASK
Casein Kinase
GHSR
DNA Methyltransferase
Ras
PD-1/PD-L1
NOS
DNA-PK
YAP
Lipase
Melatonin Receptor
Serine Protease
Aryl Hydrocarbon Receptor
Isocitrate Dehydrogenase (IDH)
DNA Alkylation
PAK
Stearoyl-CoA Desaturase (SCD)
Chk
Ephrin Receptor
IκB/IKK
NADPH-oxidase
p53
CRM1
Cholecystokinin Receptor
Vitamin
Drug Metabolite
MT Receptor
Glucosidase
Monoamine Transporter
Neuropeptide Y Receptor
FAAH
DNA
DUB
PGE Synthase
Porcupine
PAI-1
Neprilysin
Protease-activated Receptor
AhR
Monocarboxylate transporter
Amino Acids and Derivatives
IFNAR
CETP
JNK
CaSR
Liver X Receptor
Glucokinase
Annexin A
FLAP
RIP kinase
UGT
GlyT
Hexokinase
Molecular Glues
PAD
Epoxide Hydrolase
Thrombopoietin Receptor
Mucin
OXPHOS
Free radical scavengers
Sirtuin
GST
LPA Receptor
PI4K
Oxytocin Receptor
CGRP Receptor
Discoidin Domain Receptor (DDR)
NOD
S6 Kinase
NOD-like Receptor (NLR)
Melanin-concentrating Hormone Receptor (MCHR)
Advanced Glycation End Products
PROTACs
MALT
NEDD8
Ligands for Target Protein for PROTAC
Sodium-dependent phosphate transporter
Cell wall
Tie-2
TOPK
Rho
Hck
Glutaminase
IDO
SIK
IRE1
PAFR
LDL
Na-K-Cl cotransporter
Integrase
Bradykinin Receptor
Telomerase
Lipid
MNK
OAT
STING
LRRK2
Histone Acetyltransferase
GluCls
Hippo pathway
Acetyl-CoA Carboxylase
PDK
Adenosine Deaminase
SGK
Gap Junction Protein
Platelet aggregation
BMI-1
Tyrosinase
MLK
Imidazoline Receptor
Kinesin
Chloride channel
Taste receptor
GSNOR
NPC1L1
Hydrogenase
CD38
Arginase
Na+/Ca2+ Exchanger
DYRK
Necroptosis
GTPase
OCT
c-Myc
Galectin
AAK1
Neurotensin Receptor
NAMPT
PYK2
FOXO1
Prolyl Endopeptidase (PREP)
Myosin
Adiponectin Receptor
Haspin Kinase
GRK
PACAP
PROTAC Linker
HCN Channel
ACK1
Angiotensin-converting Enzyme (ACE)
Somatostatin
cAMP
ATP Citrate Lyase
Wee1
BCRP
Glutathione reductase
Survivin
GPCR19
Decarboxylase
Pyroptosis
Methionine Adenosyltransferase (MAT)
GPX
Melanocortin Receptor
CRISPR/Cas9
RXFP receptor
Anti-infection
p97
PKM

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