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Targeted Therapy Drug Library

Catalog No. L2152
  Library Compound List   Excel SDF

Targeted therapy for cancer is a treatment modality at the cellular molecular level that targets a known cancer-causing site. Common targeted drugs include small molecule drugs and monoclonal antibodies. Monoclonal antibodies have higher selectivity but are large molecule proteins, which are difficult to enter cells, and their targets are often limited to the cell surface; small molecule drugs are advantageous for targeting molecules inside tumor cells since they are small enough to easily enter tumor cells and directly target the molecules inside. With high specificity and less toxic side effects, targeted drugs have remarkable therapeutic efficacy on a variety of malignant tumors. They have become the new mainstream antitumor drugs in the last decade.

TargetMol collected 121 tumor-targeted drugs and formed the Targeted Therapy Drug Library, a powerful tool in oncotherapy research.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
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Product Description

  • 116 tumor-targeted drugs that can be used for high-throughput and high-content screening.
  • Targets include EGFR, VEGFR, c-Met, Bcr-Abl, HER2, etc.
  • All compounds have known and good biological activity, safety and bioavailability.
  • Detailed instructions, compound structures, target information, IC50 values, activity descriptions, etc.
  • Various detection techniques such as NMR, HPLC/LCMS to ensure correct structure, high purity and reduce the false-positive rates.

Library Customization

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Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L2152)

Library Composition

c-Kit (22)
VEGFR (21)
PDGFR (17)
EGFR (14)
FLT (10)
FGFR (9)
Bcr-Abl (9)
Tyrosine Kinases (6)
MEK (6)
c-RET (6)
ALK (6)
Src (6)
Raf (6)
HDAC (5)
CDK (5)
PI3K (5)
c-Met/HGFR (5)
Proteasome (4)
PARP (4)
JAK (4)
HER (4)
TAM Receptor (3)
Trk receptor (3)
Hedgehog/Smoothened (3)
Androgen Receptor (3)
Aromatase (3)
BTK (3)
CSF-1R (2)
Estrogen/progestogen Receptor (2)
IGF-1R (2)
mTOR (2)
ROS (2)
Dehydrogenase (2)
c-Fms (1)
BCL (1)
Serine Protease (1)
ROCK (1)
Retinoid Receptor (1)
Caspase (1)
GABA Receptor (1)
PPAR (1)
PKC (1)
ACK (1)
DHFR (1)
P450 (1)
Microtubule Associated (1)
Ephrin Receptor (1)
MAPK (1)
ERK (1)
Histone Methyltransferase (1)
ABC (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE