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Angiogenesis EGFR Endoxifen Z-isomer

Endoxifen Z-isomer

Catalog No. T2280   CAS 112093-28-4
Purity 99.57% Datasheet MSDS

Endoxifen (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity.

Endoxifen Z-isomer, CAS 112093-28-4
Pack Size Availability Price/USD Quantity
1 mg In stock 85.00
5 mg In stock 155.00
10 mg In stock 258.00
25 mg In stock 505.00
1 mL * 10 mM (in DMSO) In stock 155.00
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Endoxifen (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity.
Targets&IC50 ER,   ERR,   hERG Potassium Channel,   hERG,  

Description

Endoxifen (EDX) is a key active metabolite of tamoxifen (TAM) with higher affinity and specificity to estrogen receptors that also inhibits aromatase activity.

Targets&IC50

ER

ERR

hERG Potassium Channel

hERG

Synonyms
Purity 98.00%
Appearance solid
Molecular Weight 373.49
Formula C25H27NO2
CAS No. 112093-28-4

Storage

-20℃ 3 years powder

-80℃ 2 years in solvent

Solubility Information

DMSO: 10 mM

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature
1. Chae YJ, et al. Eur J Pharmacol. 2015 Apr 5;752:1-7.2. Wu X, et al. Breast Y Res. 2011 Mar 10;13(2):R27.

Related Compound Libraries

This product is contained In the following compound libraries:
Bioactive Compound Library Inhibitor Library Anti-cancer Compound Library Clinical Compound Library Endocrinology-Hormones Library Ion Channel Inhibitor Library Tyrosine kinase inhibitor library Anti-cancer Clinical Compound Library Angiogenesis related Compound Library JAK STAT Compound Library

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