Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
10 mg | 35 days | $ 78.00 | |
25 mg | 35 days | $ 175.00 | |
50 mg | 35 days | $ 250.00 | |
100 mg | 35 days | $ 460.00 |
Description | Methiothepin maleate (Metitepine) is a 5-HT1, 5-HT6, 5-HT7 serotonin receptor antagonist, which blocks serotonin autoreceptors. |
Targets&IC50 | H5-HT7 receptor:152 nM |
In vivo | The intracerebroventricular administration of aftin-4 (3–20 nmol) increased Aβ1-42, but not Aβ1-40, content in the mouse hippocampus, between 5 and 14 days after injection. Aftin-4 injection increased lipid peroxidation levels in the hippocampus, an index of oxidative stress. |
Synonyms | Metitepine |
Molecular Weight | 472.62 |
Formula | C24H28N2O4S2 |
CAS No. | 19728-88-2 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mM
You can also refer to dose conversion for different animals. More
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Methiothepin maleate 19728-88-2 GPCR/G Protein Neuroscience 5-HT Receptor Methiothepin Maleate Metitepine inhibitor inhibit