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CDK4/6-IN-8

Catalog No. T61892Cas No. 2649120-22-7

CDK4/6-IN-8 (Compound 7p) is a selective inhibitor of CDK4 with an IC50 of 5.01 nM and CDK6 with an IC50 of 3.97 nM.

CDK4/6-IN-8

CDK4/6-IN-8

Catalog No. T61892Cas No. 2649120-22-7
CDK4/6-IN-8 (Compound 7p) is a selective inhibitor of CDK4 with an IC50 of 5.01 nM and CDK6 with an IC50 of 3.97 nM.
Pack SizePriceAvailabilityQuantity
25 mg$1,5206-8 weeks
50 mg$1,9806-8 weeks
100 mg$2,5006-8 weeks
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Product Introduction

Bioactivity
Description
CDK4/6-IN-8 (Compound 7p) is a selective inhibitor of CDK4 with an IC50 of 5.01 nM and CDK6 with an IC50 of 3.97 nM.
In vitro
CDK4/6-IN-8 (Compound 7p) demonstrates anti-breast cancer activity, inhibiting MCF-7 cell viability with an IC50 of 2.8 μM over a 48-hour period at concentrations ranging from 0.1 to 656.1 μM [1].
Chemical Properties
Molecular Weight398.37
FormulaC18H18N6O5
Cas No.2649120-22-7
Storage & Solubility Information
StorageShipping with blue ice.

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