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Propiram fumarate HCl
Catalog No. T28453LCas No. 945013-73-0
Alias Propiram fumarate HCl(15686-91-6 Free base)
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
Propiram fumarate HCl
Catalog No. T28453LAlias Propiram fumarate HCl(15686-91-6 Free base)Cas No. 945013-73-0
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $195 | In Stock | |
| 5 mg | $430 | In Stock | |
| 10 mg | $636 | In Stock | |
| 25 mg | $987 | In Stock | |
| 50 mg | $1,360 | In Stock | |
| 100 mg | $1,830 | In Stock | |
| 500 mg | $3,680 | In Stock |
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Purity:99.25%
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All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.Product Introduction
Bioactivity
Chemical Properties
| Description | Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain. |
| In vivo | Propiram fumarate HCl (50 mg; single oral; 4, 6 h; 120 patients) was significantly more effective than codeine at hour 5 for Pain Intensity Difference. Propiram fumarate HCl is an effective oral analgesic similar to codeine sulfate 60 mg, with the possibility of a longer duration of action.[1] |
| Alias | Propiram fumarate HCl(15686-91-6 Free base) |
| Formula | C16H25N3O.xClH |
| Cas No. | 945013-73-0 |
Storage & Solubility Information
| Storage | Shipping with blue ice. |
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(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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