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Home > Tyrosine Kinase/Adaptors > PDGFR > Pazopanib HCl (GW786034 HCl)
Pazopanib HCl (GW786034 HCl)  
Catalog No. T6930    CAS 635702-64-6
Pack Size
Availability
Price/USD
Quantity
10mg
9 days
43.00
25mg
9 days
66.00
50mg
9 days
85.00
100mg
9 days
128.00
200mg
9 days
213.00
500mg
9 days
298.00
1g
Get quote
0.00
5g
Get quote
0.00
10mM * 1mL (in DMSO)
9 days
47.00
Bulk Size: Please Quote for Discount
Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

Pazopanib HCl (GW786034 HCl) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM in cell-free assays, respectively.

Target:
PDGFR ;
Research Area:
Others
Chemical Information:
Molecular Weight 473.98
Formula C21H23N7O2S·HCl
CAS Number 635702-64-6
Solubility DMSO: 17mg/ml(35.87 mM);Water: <1mg/ml;Ethanol: <1mg/ml
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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