Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor. Bimatoprost methyl ester is a lipophilic analog of 17-phenyl trinor PGF2α, a potent agonist for the FP receptor. 17-phenyl trinor PGF2α binds the FP receptor on ovine luteal cells with a relative potency of 756% compared to that of PGF2α. Esters of PGs serve as prodrugs, as they are efficiently hydrolyzed in certain tissues to generate the bioactive free acid.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | 4-5 weeks | $ 183.00 | |
5 mg | 4-5 weeks | $ 793.00 | |
10 mg | 4-5 weeks | $ 1,430.00 |
Description | Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor. Bimatoprost methyl ester is a lipophilic analog of 17-phenyl trinor PGF2α, a potent agonist for the FP receptor. 17-phenyl trinor PGF2α binds the FP receptor on ovine luteal cells with a relative potency of 756% compared to that of PGF2α. Esters of PGs serve as prodrugs, as they are efficiently hydrolyzed in certain tissues to generate the bioactive free acid. |
Synonyms | 17-phenyl trinor Prostaglandin F2α methyl ester |
Molecular Weight | 402.531 |
Formula | C24H34O5 |
CAS No. | 38315-47-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PBS (pH 7.2): 0.25 mg/mL
Acetonitrile: 3 mg/mL
Ethanol: 50 mg/mL
DMSO: 25 mg/mL
DMF: 25 mg/mL
You can also refer to dose conversion for different animals. More
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Bimatoprost methyl ester 38315-47-8 17-phenyl trinor Prostaglandin F2a methyl ester 17-phenyl trinor Prostaglandin F-2α methyl ester 17phenyl trinor Prostaglandin F2α methyl ester 17 phenyl trinor Prostaglandin F2α methyl ester 17-phenyl trinor Prostaglandin F2α methyl ester inhibitor inhibit