BAY-784

BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).

Catalog No. T10475Cas No. 1631164-24-3

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BAY-784

Catalog No. T10475Cas No. 1631164-24-3

BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

Pack Size	Price	Availability
25 mg	$1,520	8-10 weeks
50 mg	$1,980	8-10 weeks
100 mg	$2,500	8-10 weeks

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Product Introduction

Bioactivity

Description	BAY-784 is a gonadotropin-releasing hormone receptor (GnRH-R) antagonist (IC50s: 21 and 24 nM for human and rat GnRH-R).
Targets&IC50	GnRHR (rat):24 nM , GnRHR (human):21 nM
In vivo	BAY-784 (0.5, 3, 10, and 30 mg/kg; 24 hours; single p.o.) reduces plasma luteinizing hormone concentration in a dose-dependent manner in ovariectomized rats.

Chemical Properties

Molecular Weight	672.11
Formula	C₂₉H₂₆ClF₄N₃O₅S₂
Cas No.	1631164-24-3

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

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Keywords

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