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Boc-ypgflt(O-tbu)

Catalog No. T25168 CAS 179124-36-8

Synonyms: Boc-tyr-pro-gly-phe-leu-thr(O-t-Bu)

Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.

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Boc-ypgflt(O-tbu), CAS 179124-36-8

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.

Synonyms	Boc-tyr-pro-gly-phe-leu-thr(O-t-Bu)
Molecular Weight	853.01
Formula	C44H64N6O11
CAS No.	179124-36-8

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Rónai AZ, Magyar A, Orosz G, Borsodi A, Benyhe S, Tóth G, Makó E, Kátay E, Babka E, Medzihradszky K. Opioid antagonist properties of the highly delta-receptor-selective BOC-Tyr-Pro-Gly-Phe-Leu-Thr (OtBu) peptide and of its Phe1 and Mel1 analogues. Arch Int Pharmacodyn Ther. 1995 Nov-Dec;330(3):361-9. PubMed PMID: 8836454. 2. Makó E, Rónai AZ, Adám G, Juhász G, Ritter L, Lestár B, Crunelli V. Modulation by GABA(B) and delta opioid receptors of neurally induced responses in isolated guinea-pig taenia coli and human colonic circular muscle. J Physiol Paris. 2000 Mar-Apr;94(2):135-8. PubMed PMID: 10791695.

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Keywords

Boc-ypgflt(O-tbu) 179124-36-8 Bocypgflt(Otbu) Boc-tyr-pro-gly-phe-leu-thr(O-t-Bu) Boc ypgflt(O tbu) Inhibitor inhibitor inhibit

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