Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GNE-0439 is a novel Nav1.7-selective inhibitor (IC50: 0.34 uM) and inhibits Nav1.5 (IC50: 38.3 μM). GNE-0439 inhibits mutant N1742K channels (IC50: 0.37 uM) in membrane potential assays.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | GNE-0439 is a novel Nav1.7-selective inhibitor (IC50: 0.34 uM) and inhibits Nav1.5 (IC50: 38.3 μM). GNE-0439 inhibits mutant N1742K channels (IC50: 0.37 uM) in membrane potential assays. |
Targets&IC50 | Nav1.7:0.34 uM |
Molecular Weight | 345.48 |
Formula | C21H31NO3 |
CAS No. | 1241902-40-8 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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GNE-0439 1241902-40-8 Others GNE0439 GNE 0439 inhibitor inhibit