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CYP1B1 ligand 3

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Catalog No. T88465Cas No. 65823-65-6

CYP1B1 Ligand 3 (Compound A1) functions as a selective inhibitor of the cytochrome P450 enzyme CYP1B1, with an IC50 of 11.9 nM. It is also utilized in the synthesis of PROTAC CYP1B1 Degrader-2.

CYP1B1 ligand 3

CYP1B1 ligand 3

😃Good
Catalog No. T88465Cas No. 65823-65-6
CYP1B1 Ligand 3 (Compound A1) functions as a selective inhibitor of the cytochrome P450 enzyme CYP1B1, with an IC50 of 11.9 nM. It is also utilized in the synthesis of PROTAC CYP1B1 Degrader-2.
Pack SizePriceAvailabilityQuantity
10 mgInquiry10-14 weeks
50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
CYP1B1 Ligand 3 (Compound A1) functions as a selective inhibitor of the cytochrome P450 enzyme CYP1B1, with an IC50 of 11.9 nM. It is also utilized in the synthesis of PROTAC CYP1B1 Degrader-2.
Targets&IC50
CYP1A2:3913.5 nM, CYP1A1:278.7 nM, CYP1B1:11.9 nM
Chemical Properties
Molecular Weight369.89
FormulaC18H12ClN3S2
Cas No.65823-65-6
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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