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Home > Histone-Methyltransferase
Cat.No. Product Name Information Area
T3624 A-366 Potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50?= 3.3 n... Others
T3084 SGC707 SGC707 is a first-in-class PRMT3 chemical probe which is a potent, selective, and cel... Others
T6916 OICR-9429 OICR-9429 is a potent antagonist of the interaction of WDR5 with peptide regions of M... Others
T6900 MS023 MS023 is a potent, selective, and cell-active Type I PRMT inhibitor with IC50 of 30 n... Others
T6879 LLY-507 LLY-507 is a cell-active, potent, and selective inhibitor of protein-lysine Methyltra... Others
T6857 HLCL-61 HLCL-61 hydrochloride is a potent and selective PRMT5 inhibitor for the treatment of ... Others
T6853 GSK591 GSK591 (EPZ015866,GSK3203591) is a potent selective inhibitor of the arginine methylt... Others
T6810 CPI-360 CPI-360 is a potent, selective,and SAM-competitive EZH1 inhibitor with IC50 of 102.3 ... Others
T6809 CPI-169 CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and ... Others
T6803 Chaetocin Chaetocin, a natural product from Chaetomium species, is a histone methyltransferase ... Others
T3257 UNC0638 UNC0638 is an inhibitor of?protein lysine methyltransferases G9a(IC50<15 nM) and GLP(... Other
T3201 WDR5-0103 WDR5-0103 is a potent and selective WD repeat-containing protein 5 (WDR5) antagonist ... Cancer
T6484 EI1 EI1 is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (W... Cancer
T2649 MI-2 MI-2 (Menin-MLL Inhibitor) is a potent menin-MLL interaction inhibitor with IC50 of 4... Cancer
T2643 MI-3 MI-3 (Menin-MLL Inhibitor) is a potent menin-MLL interaction inhibitor with IC50 of 6... Cancer
T6076 EPZ015666 EPZ015666 is a potent, selective and orally bioavailable PRMT5 inhibitor with Ki of 5... Cancer
T6059 GSK343 GSK343 is a potent and selective EZH2 inhibitor with IC50 of 4 nM, showing 60 fold se... Cancer
T3099 EPZ5676 EPZ-5676 is an S-adenosyl methionine (SAM) competitive inhibitor of protein methyltra... Cancer
T3082 SGC0946 SGC0946 is a highly potent and selective DOT1L methyltransferase inhibitor with IC50 ... Cancer
T3081 EPZ004777 EPZ004777 is a potent, selective?DOT1L?inhibitor with?IC50?of 0.4 nM. Cancer
T3057 UNC1999 UNC1999 is a potent, orally bioavailable and selective inhibitor of EZH2 and EZH1 wit... Cancer
T2435 EPZ011989 EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM fo... Cancer
T2354 UNC 0631 UNC0631 is a potent histone methyltransferase G9a inhibitor with IC50 of 4 nM. Other
T2352 AMI-1 AMI-1 is a potent and specific Histone Methyltransferase (HMT) inhibitor with IC50 of... Other
T2216 Entacapone Entacapone is a selective, reversible catechol-O-methyl transferase (COMT) inhibitor ... Nervous system
T2097 C7280948 C-7280948 is a PRMT1 inhibitor. Other
T2079 GSK126 GSK126 is a potent, highly selective EZH2 methyltransferase inhibitor with IC50 of 9.... Other
T2038 RG108 RG108 is an inhibitor of DNA methyltransferase with IC50 of 115 nM in a cell-free ass... Other
T1987 PFI-2 PFI-2 is a potent, selective, and cell-active lysine methyltransferase SETD7 inhibito... Other
T1959 BIX 01294 Trihydrochloride BIX01294 is an inhibitor of G9a histone methyltransferase with IC50 of 2.7 μM in a ce... Other