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TargetMol | Compound Library

Highly Selective Inhibitor Library

Catalog No. L2010

Highly selective inhibitors are able to specifically interact with the targeted molecule or pathway selectively with relatively little effect on other non-targeted molecules or pathway. The advantage of highly selective inhibitors over non-selective inhibitors is that they act more precisely on the target, thereby reducing interference with non-targets and reducing possible side-effects and toxicity. Highly selective inhibitors are widely used in drug development, especially in the treatment of cancer and other complex diseases, and are applied to intervene more effectively in pathological processes, improve the effectiveness of treatment, and reduce the incidence of adverse effects. TargetMol has collected 575 highly selective inhibitors, the vast majority of which are at least a hundred times more selective relative to other targets, making the Highly Selective Inhibitor Library an effective tool for drug development.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2010

Highly Selective Inhibitor Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Product Description Product Description

  • A collection of 575 highly selective inhibitors;
  • Covering 170 drug targets;
  • Some inhibitors have been approved by FDA;
  • Covering a variety of signaling pathways, such as ion channels; NF-κB; PI3K/Akt/mTOR signaling; MAPK and so on.
  • Diverse structure, strong biological activity, cell penetrable;
  • Detailed specifications, compound structure, target information, IC50 value, activity description, etc;
  • NMR, HPLC/LCMS and other detection techniques to ensure the correct structure, high purity of the product and to reduce false positives.

Packaging And Storage | TargetMol Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
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Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
EGFR
PI3K
Histone Methyltransferase
Epigenetic Reader Domain
CDK
BTK
mTOR
c-Met/HGFR
GSK-3
Proteasome
Aurora Kinase
FGFR
DPP-4
Src
Raf
HDAC
MEK
JAK
PDGFR
Antibacterial
FLT
PARP
VEGFR
HIV Protease
Chk
COX
SGLT
Cysteine Protease
TRP/TRPV Channel
ERK
PDE
BCL
PLK
Antibiotic
DNA-PK
Histone Demethylase
PPAR
TGF-beta/Smad
DNA/RNA Synthesis
SARS-CoV
Trk receptor
IκB/IKK
ATM/ATR
HER
p38 MAPK
Dehydrogenase
Ferroptosis
Phosphatase
Mitophagy
Virus Protease
Serine Protease
PKC
Adrenergic Receptor
MMP
Histone Acetyltransferase
ALK
c-Fms
P450
c-Kit
Ras
Ligands for Target Protein for PROTAC
PERK
Lipase
PKA
Tyrosine Kinases
Wnt/beta-catenin
ROCK
MAO
CSF-1R
RIP kinase
FAAH
DUB
Akt
Sirtuin
Casein Kinase
GPR
PDK
5-HT Receptor
Potassium Channel
AChR
TAM Receptor
HCV Protease
RAAS
JNK
Factor Xa
Serine/threonin kinase
Caspase
iGluR
E1/E2/E3 Enzyme
GluR
IGF-1R
MNK
HSP
Prostaglandin Receptor
Influenza Virus
STAT
Syk
S6 Kinase
Thrombin
Monoamine Oxidase
Kinesin
Proton pump
NOS
Dopamine Receptor
Estrogen/progestogen Receptor
LPL Receptor
Adenosine Receptor
DYRK
NADPH
Glutathione Peroxidase
Tie-2
Estrogen Receptor/ERR
Parasite
Pim
IDO
Bcr-Abl
GRK
Phosphorylase
Mitochondrial Metabolism
Isocitrate Dehydrogenase (IDH)
Integrase
Reactive Oxygen Species
HSV
CXCR
Endothelin Receptor
KSP
cAMP
CaMK
Indoleamine 2,3-Dioxygenase (IDO)
MAPK
LRRK2
transporter
AMPK
Hydroxylase
Cannabinoid Receptor
Neurokinin receptor
NOD
Sodium Channel
NOD-like Receptor (NLR)
Mdm2
ATPase
Chloride channel
Carbonic Anhydrase
Transferase
MALT
Dynamin
YAP
Antifungal
IFNAR
Histamine Receptor
Progesterone Receptor
Galectin
Rho
NAMPT
Glutaminase
Calcium Channel
Immunology/Inflammation related
Glucocorticoid Receptor
SIK
Topoisomerase
IRE1
MTH1
FABP
NMDAR
GlyT
Monoamine Transporter
ROS
Opioid Receptor
Neuropeptide Y Receptor
Fatty Acid Synthase
PAK
CCR
Vasopressin Receptor
OX Receptor
Epoxide Hydrolase
ACK
Lipoxygenase
DNA
Interleukin
Telomerase
Wee1
BCRP
AChE
P-gp
Porcupine
TLR
CD73
Decarboxylase
cGAS
ASK
Reverse Transcriptase
LPA Receptor
NF-κB
Phospholipase
GABA Receptor
HIF
c-RET
SGK
Complement System
DAPK
Platelet aggregation
DNA Methyltransferase
BMI-1
IRAK
Sigma receptor
Microtubule Associated
Protease-activated Receptor
FAK
HIF/HIF Prolyl-Hydroxylase
MLK
PD-1/PD-L1
NO Synthase
PKM
S1P Receptor

Keywords