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(3S,4S)-PF-06459988

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Catalog No. T39299Cas No. 1858291-14-1

(3S, 4S)-PF-06459988 is the less active S enantiomer of PF-06459988, a potent irreversible inhibitor of T790M mutant epidermal growth factor receptor (EGFR), exhibiting excellent selectivity against EGFR wild-type due to its minimally reactive electrophile, reducing off-target labeling likelihood.

(3S,4S)-PF-06459988
Other Forms of (3S,4S)-PF-06459988:
PF-06459988T164921428774-45-1
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(3S,4S)-PF-06459988

😃Good
Catalog No. T39299Cas No. 1858291-14-1
(3S, 4S)-PF-06459988 is the less active S enantiomer of PF-06459988, a potent irreversible inhibitor of T790M mutant epidermal growth factor receptor (EGFR), exhibiting excellent selectivity against EGFR wild-type due to its minimally reactive electrophile, reducing off-target labeling likelihood.
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2 mg$825 days
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Product Introduction

Bioactivity
Description
(3S, 4S)-PF-06459988 is the less active S enantiomer of PF-06459988, a potent irreversible inhibitor of T790M mutant epidermal growth factor receptor (EGFR), exhibiting excellent selectivity against EGFR wild-type due to its minimally reactive electrophile, reducing off-target labeling likelihood.
Chemical Properties
Molecular Weight431.88
FormulaC19H22ClN7O3
Cas No.1858291-14-1
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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Keywords

(3S,4S)PF06459988PF 06459988(3S,4S) PF 06459988PF-06459988PF06459988
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