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(Rac)-PF-06250112

Name: (Rac)-PF-06250112
Brand: TargetMol
SKU: T12673
Rating: 4.5 (1 reviews)

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Catalog No. T12673Cas No. 1609465-88-4

(Rac)-PF-06250112 is a racemic form of PF-06250112, a potent and highly selective BTK inhibitor that is orally bioavailable; it also inhibits BMX non-receptor tyrosine kinase and TEC [1].

(Rac)-PF-06250112

😃Good

Catalog No. T12673Cas No. 1609465-88-4

(Rac)-PF-06250112 is a racemic form of PF-06250112, a potent and highly selective BTK inhibitor that is orally bioavailable; it also inhibits BMX non-receptor tyrosine kinase and TEC [1].

Pack Size	Price	Availability
25 mg	$1,520	8-10 weeks
50 mg	$1,980	8-10 weeks
100 mg	$2,500	8-10 weeks

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Product Introduction

Bioactivity

Description

(Rac)-PF-06250112 is a racemic form of PF-06250112, a potent and highly selective BTK inhibitor that is orally bioavailable; it also inhibits BMX non-receptor tyrosine kinase and TEC [1].

Chemical Properties

Molecular Weight	438.43
Formula	C₂₂H₂₀F₂N₆O₂
Cas No.	1609465-88-4
Relative Density.	1.46 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 250 mg/mL (570.22 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.2809 mL	11.4043 mL	22.8087 mL	114.0433 mL
5 mM	0.4562 mL	2.2809 mL	4.5617 mL	22.8087 mL
10 mM	0.2281 mL	1.1404 mL	2.2809 mL	11.4043 mL
20 mM	0.1140 mL	0.5702 mL	1.1404 mL	5.7022 mL
50 mM	0.0456 mL	0.2281 mL	0.4562 mL	2.2809 mL
100 mM	0.0228 mL	0.1140 mL	0.2281 mL	1.1404 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

PF 06250112PF06250112(Rac)PF06250112PF-06250112(Rac) PF 06250112