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ARL67156 trisodium salt

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ARL67156 trisodium salt

Catalog No. T14320Cas No. 1021868-83-6

ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. ARL67156 trisodium salt is an inhibitor of ecto-ATPase.

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Pack Size	Price	Availability	Quantity
10 mg	$755	35 days

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Product Introduction

Bioactivity

Description	ARL 67156 is a weak competitive inhibitor of NTPDase1 (CD39), NTPDase3 and NPP1, with Kis of 11, 18 and 12 μM, respectively[1]. ARL67156 trisodium salt is an inhibitor of ecto-ATPase.
In vitro	ARL67156 does not significantly inhibit the activity of NTPDase2, NTPDase8, NPP3, and ecto-5′-nucleotidase (CD73), yet it diminishes their activity [1]. In addition, the trisodium salt form of ARL67156 effectively impedes UTP breakdown in superior cervical ganglion cells and enhances contractions triggered by this nucleotide in isolated rat tail artery.

Chemical Properties

Molecular Weight	788.079
Formula	C15H24Br2N5Na3O12P3
Cas No.	1021868-83-6

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 25 mg/mL (31.72 mM), Sonication is recommended.

Solution Preparation Table

H2O

	1mg	5mg	10mg	50mg
50 mM	0.0254 mL	0.1269 mL	0.2538 mL	1.2689 mL
100 mM	0.0127 mL	0.0634 mL	0.1269 mL	0.6345 mL

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Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

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Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

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