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Pack Size | Price | Availability | Quantity |
---|---|---|---|
5 mg | $364 | 6-8 weeks | |
25 mg | $1,450 | 6-8 weeks | |
50 mg | $1,890 | 6-8 weeks | |
100 mg | $2,800 | 6-8 weeks |
Description | SK1-IN-1 is a potent inhibitor of sphingosine kinase 1 (SPHK1)(IC50 of 58 nM). |
In vivo | SK1-IN-1 exhibits a considerable enhancement in intrinsic clearance, especially when assessed against human liver microsomes. Chosen for rat pharmacokinetic (PK) studies, it reveals moderate oral bioavailability alongside acceptable circulation half-lives. |
Molecular Weight | 398.5 |
Formula | C22H30N4O3 |
Cas No. | 1218816-71-7 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | |||||||||||||||||||||||||||||||||||
Solubility Information | DMSO: 100 mg/mL (250.94 mM) | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
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