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AMXI-5001

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Catalog No. T62847Cas No. 2170491-77-5

AMXI-5001 is a potent, orally active inhibitor of PARP1/2 and microtubule aggregation. AMXI-5001 shows selective anti-tumor cytotoxicity against a wide range of human cancer cells with IC50s well below those of existing clinical PARP1/2 inhibitors and induces complete regression of established tumors, including very large ones.

AMXI-5001
Other Forms of AMXI-5001:
AMXI-5001 hydrochlorideT63328
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AMXI-5001

😃Good
Catalog No. T62847Cas No. 2170491-77-5
AMXI-5001 is a potent, orally active inhibitor of PARP1/2 and microtubule aggregation. AMXI-5001 shows selective anti-tumor cytotoxicity against a wide range of human cancer cells with IC50s well below those of existing clinical PARP1/2 inhibitors and induces complete regression of established tumors, including very large ones.
Pack SizePriceAvailabilityQuantity
25 mg$1,6206-8 weeks
50 mg$2,1106-8 weeks
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Product Introduction

Bioactivity
Description
AMXI-5001 is a potent, orally active inhibitor of PARP1/2 and microtubule aggregation. AMXI-5001 shows selective anti-tumor cytotoxicity against a wide range of human cancer cells with IC50s well below those of existing clinical PARP1/2 inhibitors and induces complete regression of established tumors, including very large ones.
Chemical Properties
Molecular Weight457.46
FormulaC25H20FN5O3
Cas No.2170491-77-5
Storage & Solubility Information
StorageShipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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