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CAY10727 is an inhibitor of protein arginine deiminase 3 (PAD3; kinact/KI= 15,600 M-1min-1).1It is selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
100 μg | $429 | 35 days | |
250 μg | $932 | 35 days | |
500 μg | $1,730 | 35 days | |
1 mg | $2,970 | 35 days |
Description | CAY10727 is an inhibitor of protein arginine deiminase 3 (PAD3; kinact/KI= 15,600 M-1min-1).1It is selective for PAD3 over PAD1, -2, and -4 (kinact/KIs = 360, 1,110, and 1,460 M-1min-1, respectively). 1.Jamali, H., Khan, H.A., Stringer, J.R., et al.Identification of multiple structurally distinct, nonpeptidic small molecule inhibitors of protein arginine deiminase 3 using a substrate-based fragment methodJ. Am. Chem. Soc.137(10)3616-3621(2015) |
Molecular Weight | 433.33 |
Formula | C21H22Cl2N4O2 |
Cas No. | 1671088-84-8 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. | ||||||||||||||||||||||||||||||
Solubility Information | DMF: 30 mg/mL (69.23 mM), Sonication is recommended. DMSO: 30 mg/mL (69.23 mM), Sonication is recommended. DMSO:PBS (pH 7.2) (1:1): 0.5 mg/mL (1.15 mM), Sonication is recommended. Ethanol: 10 mg/mL (23.08 mM), Sonication is recommended. | ||||||||||||||||||||||||||||||
Solution Preparation Table | |||||||||||||||||||||||||||||||
Ethanol/DMF/DMSO
DMF/DMSO
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