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CDK12-IN-7

Catalog No. T88012Cas No. 3033863-94-1

CDK12-IN-7 (Compound 2), a dual inhibitor of CDK12 and CDK2, exhibits IC 50 values of 42 nM and 196 nM, respectively. This compound demonstrates anti-cell proliferation properties, making it applicable in cancer research.

CDK12-IN-7

CDK12-IN-7

Catalog No. T88012Cas No. 3033863-94-1
CDK12-IN-7 (Compound 2), a dual inhibitor of CDK12 and CDK2, exhibits IC 50 values of 42 nM and 196 nM, respectively. This compound demonstrates anti-cell proliferation properties, making it applicable in cancer research.
Pack SizePriceAvailabilityQuantity
10 mgInquiry10-14 weeks
50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
CDK12-IN-7 (Compound 2), a dual inhibitor of CDK12 and CDK2, exhibits IC 50 values of 42 nM and 196 nM, respectively. This compound demonstrates anti-cell proliferation properties, making it applicable in cancer research.
Targets&IC50
CDK2:196 nM, CDK12:42 nM
In vitro
CDK12-IN-7 inhibits the proliferation of A2780 cells, with an IC50 value of 429 nM [1].
Chemical Properties
Molecular Weight663.65
FormulaC32H32F3N9O4
Cas No.3033863-94-1
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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