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EF-4-177

Catalog No. T88162Cas No. 2891574-93-7

EF-4-177, an orally active, allosteric CDK2 inhibitor, exhibits an IC50 value of 87 nM. It has been shown to disrupt spermatogenesis.

EF-4-177

EF-4-177

Catalog No. T88162Cas No. 2891574-93-7
EF-4-177, an orally active, allosteric CDK2 inhibitor, exhibits an IC50 value of 87 nM. It has been shown to disrupt spermatogenesis.
Pack SizePriceAvailabilityQuantity
10 mgInquiry10-14 weeks
50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
EF-4-177, an orally active, allosteric CDK2 inhibitor, exhibits an IC50 value of 87 nM. It has been shown to disrupt spermatogenesis.
Targets&IC50
CDK2/cyclinE:87 nM
Chemical Properties
Molecular Weight431.38
FormulaC18H14F5N3O2S
Cas No.2891574-93-7
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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