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Emicerfont

Name: Emicerfont
Brand: TargetMol
SKU: T15214
Price: 28 EUR
Availability: InStock
Rating: 4.5 (1 reviews)

Catalog No. T15214Cas No. 786701-13-1

Alias GW876008

Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).

Emicerfont

Catalog No. T15214Alias GW876008Cas No. 786701-13-1

Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).

Pack Size	Price	Availability
25 mg	$1,970	8-10 weeks
50 mg	$2,580	8-10 weeks
100 mg	$3,400	8-10 weeks

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Product Introduction

Bioactivity

Description	Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).
Targets&IC50	CRF1 receptor:66 nM
In vivo	Emicerfont (10 mg/kg) treatment, decreases i.c.v. CRF-induced gerbil forepaw treading and marmoset defensive postures. Emicerfont (30 mg/kg) treatment, also reduces rat pup ultrasonic vocalization.
Alias	GW876008

Chemical Properties

Molecular Weight	404.46
Formula	C₂₂H₂₄N₆O₂
Cas No.	786701-13-1

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

GW-876008EmicerfontGW 876008