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Gefitinib-d8

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Catalog No. T11384Cas No. 857091-32-8
Alias ZD1839 D8, Gefitinib D8

Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells. Gefitinib D8 is a deuterium labeled Gefitinib.

Gefitinib-d8
Other Forms of Gefitinib-d8:

Gefitinib-d8

😃Good
Catalog No. T11384Alias ZD1839 D8, Gefitinib D8Cas No. 857091-32-8
Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells. Gefitinib D8 is a deuterium labeled Gefitinib.
Pack SizePriceAvailabilityQuantity
1 mg$1727-10 days
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Product Introduction

Bioactivity
Description
Gefitinib is an EGFR tyrosine kinase inhibitor, with IC50 of 2-37 nM in NR6wtEGFR cells. Gefitinib D8 is a deuterium labeled Gefitinib.
Targets&IC50
Tyr992 site (NR6wtEGFR cells):37 nM , Tyr1173 site (NR6wtEGFR cells):37 nM
AliasZD1839 D8, Gefitinib D8
Chemical Properties
Molecular Weight454.95
FormulaC22H24ClFN4O3
Cas No.857091-32-8
Relative Density.no data available
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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Keywords

Tyr992 site, in NR6wtEGFR cellsTyr1173 site, in NR6wtEGFR cellsGefitinib-d-8Gefitinib-d8Gefitinibd8
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