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GPR30 agonist-1
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Catalog No. T40517Cas No. 415919-74-3
Alias GPR30 agonist-1
GPR30 agonist-1 is a compound that acts as an agonist for G protein-coupled receptor 30 (GPR30), inducing vasorelaxation.
GPR30 agonist-1
😃Good
Catalog No. T40517Alias GPR30 agonist-1Cas No. 415919-74-3
GPR30 agonist-1 is a compound that acts as an agonist for G protein-coupled receptor 30 (GPR30), inducing vasorelaxation.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 2 mg | $73 | 5 days |
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Product Introduction
Bioactivity
Chemical Properties
| Description | GPR30 agonist-1 is a compound that acts as an agonist for G protein-coupled receptor 30 (GPR30), inducing vasorelaxation. |
| In vivo | GPR30 agonist-1 (compound 5408-0877) induces a concentration-dependent relaxation in carotid arteries of both male and female rats at concentrations from 1 nM to 10 μM. This effect is abolished by the removal of the endothelium and inhibited by the nitric oxide synthase inhibitor NG-nitro-l-arginine methyl ester (100 μM). |
| Alias | GPR30 agonist-1 |
| Molecular Weight | 374.253 |
| Formula | C19H17BrFNO |
| Cas No. | 415919-74-3 |
| Relative Density. | 1.394 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc
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