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JTP-117968

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Catalog No. T63636Cas No. 2250132-99-9

JTP-117968 is a selective glucocorticoid receptor modulator (non-steroidal SGRM with an IC50 value of 6.8 nM) that exhibits improved transcriptional inhibition/transactivation dissociation.

JTP-117968

JTP-117968

😃Good
Catalog No. T63636Cas No. 2250132-99-9
JTP-117968 is a selective glucocorticoid receptor modulator (non-steroidal SGRM with an IC50 value of 6.8 nM) that exhibits improved transcriptional inhibition/transactivation dissociation.
Pack SizePriceAvailabilityQuantity
25 mg$1,520 10-14 weeks
50 mg$1,980 10-14 weeks
100 mg$2,500 10-14 weeks
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Product Introduction

Bioactivity
Description
JTP-117968 is a selective glucocorticoid receptor modulator (non-steroidal SGRM with an IC50 value of 6.8 nM) that exhibits improved transcriptional inhibition/transactivation dissociation.
Chemical Properties
Molecular Weight520.59
FormulaC31H31F3N2O2
Cas No.2250132-99-9
Storage & Solubility Information
StorageShipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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