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LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM).
Pack Size | Price | Availability | Quantity |
---|---|---|---|
25 mg | $2,420 | 10-14 weeks | |
50 mg | $3,180 | 10-14 weeks | |
100 mg | $4,300 | 10-14 weeks |
Description | LTD4 antagonist 1 is a potent and orally active antagonist of leukotriene D4 (LTD4; Ki: 0.57 nM). |
Targets&IC50 | LTD4:0.57 nM (ki) |
In vitro | LTD4 antagonist 1 (Compound 38b) shows a Ki of 0.57 nM for the displacement of [3H]LTD4 on guinea pig lung membranes, a pKB of 9.93 versus LTE4 on guinea pig trachea. |
In vivo | LTD4 antagonist 1 shows a ED50 (i.v.)/ED50 (p.o.) of 0.036 and 1.44 μmol/kg in LTD4-induced bronchoconstriction in guinea pigs. |
Molecular Weight | 615.66 |
Formula | C31H32F3N3O5S |
Cas No. | 136564-67-5 |
Relative Density. | no data available |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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