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LUF5771

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Catalog No. T61307Cas No. 1141802-49-4

LUF5771 is a highly potent allosteric inhibitor of recombinant luteinizing hormone (recLH) and Org 43553. It exhibits partial activation of the LH receptor with low efficacy [1].

LUF5771

LUF5771

😃Good
Catalog No. T61307Cas No. 1141802-49-4
LUF5771 is a highly potent allosteric inhibitor of recombinant luteinizing hormone (recLH) and Org 43553. It exhibits partial activation of the LH receptor with low efficacy [1].
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2 mg$585 days
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Product Introduction

Bioactivity
Description
LUF5771 is a highly potent allosteric inhibitor of recombinant luteinizing hormone (recLH) and Org 43553. It exhibits partial activation of the LH receptor with low efficacy [1].
In vitro
LUF5771 (1 μM or 10 μM) allosteric inhibition is concentration-dependent. LUF5771 significantly increases radioligand dissociation. LUF5771 probably binds to the seven transmembrane domain like Org 43553 does. LUF5771 (10 μM) alone is able to partially activate the LH receptor by 31±4% [1].
Chemical Properties
Molecular Weight357.44
FormulaC24H23NO2
Cas No.1141802-49-4
Storage & Solubility Information
StorageShipping with blue ice.

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