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MRK-898, an orally active modulator of the GABA(A) receptor, selectively interacts with the α1, α2, α3, and α5 subunits, displaying K i values of 1.2 nM, 1.0 nM, 0.73 nM, and 0.50 nM, respectively. It is noteworthy that the α1-containing receptors of GABA(A) are classified as "sedative," whereas receptors containing α2 and/or α3 are designated as "anxiolytic" subtype(s) [1].
Pack Size | Price | Availability | Quantity |
---|---|---|---|
10 mg | Inquiry | 10-14 weeks | |
50 mg | Inquiry | 10-14 weeks |
Description | MRK-898, an orally active modulator of the GABA(A) receptor, selectively interacts with the α1, α2, α3, and α5 subunits, displaying K i values of 1.2 nM, 1.0 nM, 0.73 nM, and 0.50 nM, respectively. It is noteworthy that the α1-containing receptors of GABA(A) are classified as "sedative," whereas receptors containing α2 and/or α3 are designated as "anxiolytic" subtype(s) [1]. |
Targets&IC50 | α2 GABA(A) receptor:1.0 nM (Ki), α1 GABA(A) receptor:1.2 nM (Ki), α3 GABA(A) receptor:0.73 nM (Ki) |
Molecular Weight | 400.3 |
Formula | C20H9F5N4 |
Cas No. | 461450-30-6 |
Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
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