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PMX-53

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Catalog No. T28429Cas No. 219639-75-5
Alias PMX53, PMX 53

PMX-53 is a Mas-related gene 2 (MrgX2) agonist and C5aR(CD88) antagonist. PMX-53 reduces atherosclerotic lesions in a mouse model of atherosclerosis, inhibits lung metastasis in a mouse breast cancer model, inhibits C5a-induced hypernociception in rats.

PMX-53
Other Forms of PMX-53:

PMX-53

😃Good
Catalog No. T28429Alias PMX53, PMX 53Cas No. 219639-75-5
PMX-53 is a Mas-related gene 2 (MrgX2) agonist and C5aR(CD88) antagonist. PMX-53 reduces atherosclerotic lesions in a mouse model of atherosclerosis, inhibits lung metastasis in a mouse breast cancer model, inhibits C5a-induced hypernociception in rats.
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1 mg$77535 days
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Product Introduction

Bioactivity
Description
PMX-53 is a Mas-related gene 2 (MrgX2) agonist and C5aR(CD88) antagonist. PMX-53 reduces atherosclerotic lesions in a mouse model of atherosclerosis, inhibits lung metastasis in a mouse breast cancer model, inhibits C5a-induced hypernociception in rats.
Targets&IC50
C5aR:20 nM (IC50)
AliasPMX53, PMX 53
Chemical Properties
Molecular Weight896.09
FormulaC47H65N11O7
Cas No.219639-75-5
Relative Density.1.40 g/cm3 (Predicted)
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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PMX-53
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