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PROTAC ERα Degrader-10

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Catalog No. T203319Cas No. 2421260-43-5

PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.

PROTAC ERα Degrader-10

PROTAC ERα Degrader-10

😃Good
Catalog No. T203319Cas No. 2421260-43-5
PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.
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Product Introduction

Bioactivity
Description
PROTACERα Degrader-10 (Compound 160a) is an orally bioavailable ERα degrader with a DC50 of 0.37-1.1 nM in MCF7, T47D, and CAMA-1 cells. It demonstrates antitumor activity in mouse models.
Chemical Properties
Molecular Weight723.9
FormulaC45H49N5O4
Cas No.2421260-43-5
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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