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S16–1029
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S16–1029

S16–1029
S16–1029 is a selective, orally active butyrylcholinesterase (BChE) inhibitor with IC50 values of 11.35 nM for eqBChE and 48.1 nM for hBChE. It can cross the blood-brain barrier (BBB) and reach the central nervous system (CNS), making it suitable for Alzheimer's disease (AD) research [1].
Catalog No. T87351Cas No. 2653349-51-8
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S16–1029

Catalog No. T87351Cas No. 2653349-51-8
S16–1029 is a selective, orally active butyrylcholinesterase (BChE) inhibitor with IC50 values of 11.35 nM for eqBChE and 48.1 nM for hBChE. It can cross the blood-brain barrier (BBB) and reach the central nervous system (CNS), making it suitable for Alzheimer's disease (AD) research [1].
All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.
Pack SizePriceAvailabilityQuantity
10 mgInquiry10-14 weeks
50 mgInquiry10-14 weeks
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Product Introduction

Bioactivity
Description
S16–1029 is a selective, orally active butyrylcholinesterase (BChE) inhibitor with IC50 values of 11.35 nM for eqBChE and 48.1 nM for hBChE. It can cross the blood-brain barrier (BBB) and reach the central nervous system (CNS), making it suitable for Alzheimer's disease (AD) research [1].
Targets&IC50
eqBCHE:11.35 nM, hBCHE:48.1 nM
Chemical Properties
Molecular Weight447.49
FormulaC23H25N7O3
Cas No.2653349-51-8
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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