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TMX-2164

Catalog No. T67949Cas No. 2418022-85-0

TMX-2164, a potent and irreversible inhibitor of B-cell lymphoma 6 (BCL6), demonstrates an IC50 of 152 nM, indicating strong inhibitory efficacy. It exhibits prolonged target engagement and effectively inhibits cell proliferation.

TMX-2164

TMX-2164

Catalog No. T67949Cas No. 2418022-85-0
TMX-2164, a potent and irreversible inhibitor of B-cell lymphoma 6 (BCL6), demonstrates an IC50 of 152 nM, indicating strong inhibitory efficacy. It exhibits prolonged target engagement and effectively inhibits cell proliferation.
Pack SizePriceAvailabilityQuantity
25 mg$1,8208-10 weeks
50 mg$2,3808-10 weeks
100 mg$3,1008-10 weeks
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Product Introduction

Bioactivity
Description
TMX-2164, a potent and irreversible inhibitor of B-cell lymphoma 6 (BCL6), demonstrates an IC50 of 152 nM, indicating strong inhibitory efficacy. It exhibits prolonged target engagement and effectively inhibits cell proliferation.
In vitro
2-heptyl-3-hydroxy-4(1H)-Quinolone (60 µM) increases secretion of the metabolite pyocyanin and the lectin PA-IL, as well as increases biofilm production in P. aeruginosa populations.[2]
2-heptyl-3-hydroxy-4(1H)-Quinolone (40 µM) reduces iron levels in P. aeruginosa growth media when used at a concentration and acts as an iron chelator in a Fe(III)-sulfate solution.[3]
Chemical Properties
Molecular Weight591.01
FormulaC25H24ClFN6O6S
Cas No.2418022-85-0
Storage & Solubility Information
StorageShipping with blue ice.

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