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TOP1288

Catalog No. T87546Cas No. 1630202-02-6

TOP1288 is a narrow-spectrum kinase inhibitor targeting P38α, Src, and Syk kinases, with IC 50 values of 116nM, 24nM, and 659nM, respectively. It effectively inhibits inflammatory cytokine release from inflamed biopsies and myofibroblasts [1].

TOP1288

TOP1288

Catalog No. T87546Cas No. 1630202-02-6
TOP1288 is a narrow-spectrum kinase inhibitor targeting P38α, Src, and Syk kinases, with IC 50 values of 116nM, 24nM, and 659nM, respectively. It effectively inhibits inflammatory cytokine release from inflamed biopsies and myofibroblasts [1].
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Product Introduction

Bioactivity
Description
TOP1288 is a narrow-spectrum kinase inhibitor targeting P38α, Src, and Syk kinases, with IC 50 values of 116nM, 24nM, and 659nM, respectively. It effectively inhibits inflammatory cytokine release from inflamed biopsies and myofibroblasts [1].
Chemical Properties
Molecular Weight839.96
FormulaC43H49N7O9S
Cas No.1630202-02-6
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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