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(Rac)-CP-601927 hydrochloride

Catalog No. T39833Cas No. 230615-01-7

(Rac)-CP-601927 hydrochloride is the racemate form of CP-601927, a nicotinic acetylcholine receptor (nAChR) agonist, with Ki values of 1.2 nM for α4β2 and 102 nM for α3β4 nAChR.

(Rac)-CP-601927 hydrochloride
Other Forms of (Rac)-CP-601927 hydrochloride:
CP-601927T31066357425-02-6
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(Rac)-CP-601927 hydrochloride

Catalog No. T39833Cas No. 230615-01-7
(Rac)-CP-601927 hydrochloride is the racemate form of CP-601927, a nicotinic acetylcholine receptor (nAChR) agonist, with Ki values of 1.2 nM for α4β2 and 102 nM for α3β4 nAChR.
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Product Introduction

Bioactivity
Description
(Rac)-CP-601927 hydrochloride is the racemate form of CP-601927, a nicotinic acetylcholine receptor (nAChR) agonist, with Ki values of 1.2 nM for α4β2 and 102 nM for α3β4 nAChR.
In vitro
CP-601927 has been shown to elicit notable antidepressant-like effects in mice. It achieves this by either decreasing cholinergic signaling through diminished efficacy or by desensitizing α4β2* nAChRs[1].
Chemical Properties
Molecular Weight263.69
FormulaC12H13ClF3N
Cas No.230615-01-7
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Keywords

CP 601927 HydrochlorideCP601927 Hydrochloride(Rac)CP601927 hydrochlorideCP-601927 Hydrochloride(Rac) CP 601927 hydrochloride
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