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(rel)-PROTAC ERRα Degrader-1

Catalog No. T18651

(rel)-PROTAC ERRα Degrader-1 is a relative configuration of PROTAC ERRα Degrader-1, which is an estrogen-related receptor alpha (ERRa) degrader. PROTAC ERRα Degrader-1 consists of an MDM2 ligand binding moiety, a linker and an ERRa binding moiety [1].

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Pack Size	Price	Availability	Quantity
100 mg	Inquiry	Backorder
500 mg	Inquiry	Backorder

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Product Introduction

Bioactivity

Description

Chemical Properties

Molecular Weight	1108.91
Formula	C54H49Cl2F6N7O8
Cas No.

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 100 mg/mL (90.18 mM)

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	0.9018 mL	4.5089 mL	9.0179 mL	45.0893 mL
5 mM	0.1804 mL	0.9018 mL	1.8036 mL	9.0179 mL
10 mM	0.0902 mL	0.4509 mL	0.9018 mL	4.5089 mL
20 mM	0.0451 mL	0.2254 mL	0.4509 mL	2.2545 mL
50 mM	0.0180 mL	0.0902 mL	0.1804 mL	0.9018 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

Dose Conversion

You can also refer to dose conversion for different animals. More

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc

Keywords

(rel)-PROTAC ERRa Degrader-1(rel)-PROTAC ERRα Degrader-1(rel)PROTAC ERRα Degrader1(rel) PROTAC ERRα Degrader 1(rel)-PROTAC ERRalpha Degrader-1