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α-2,3-sialyltransferase-IN-1

Name: α-2,3-sialyltransferase-IN-1
Brand: TargetMol
SKU: T13429
Rating: 4.5 (1 reviews)

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Catalog No. T13429Cas No. 881179-06-2

Alias Lith-O-Asp analog

α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is an α-2,3-sialyltransferase inhibitor with anticancer activity. Vapendavir diphosphate inhibits EV71 replication.

α-2,3-sialyltransferase-IN-1

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Purity: 98%

Catalog No. T13429Alias Lith-O-Asp analogCas No. 881179-06-2

α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is an α-2,3-sialyltransferase inhibitor with anticancer activity. Vapendavir diphosphate inhibits EV71 replication.

Pack Size	Price	Availability
25 mg	$1,520	6-8 weeks
50 mg	$1,980	6-8 weeks
100 mg	$2,500	6-8 weeks

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Purity:98%

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COA

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Product Introduction

Bioactivity

Description	α-2,3-sialyltransferase-IN-1 (Lith-O-Asp analog) is an α-2,3-sialyltransferase inhibitor with anticancer activity. Vapendavir diphosphate inhibits EV71 replication.
Targets&IC50	α-2,3-sialyltransferase:6 μM
In vitro	α-2,3-sialyltransferase-IN-1 is a non-competitive inhibitor of α-2,3-sialyltransferase with an IC50 value of 6 μM. α-2,3-sialyltransferase-IN-1 is compound 17 in the reference. [1]
Alias	Lith-O-Asp analog

Chemical Properties

Molecular Weight	491.66
Formula	C₂₈H₄₅NO₆
Cas No.	881179-06-2
Smiles	C[C@@]12[C@]([C@]3([C@@]([C@]4(C)[C@](CC3)(C[C@H](OC([C@@H](CC(O)=O)N)=O)CC4)[H])(CC1)[H])[H])(CC[C@@]2([C@@H](CCC(O)=O)C)[H])[H]
Relative Density.	1.19 g/cm3 (Predicted)

Storage & Solubility Information

Storage

store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

Solubility Information

DMSO: 80 mg/mL (162.71 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0339 mL	10.1696 mL	20.3393 mL	101.6963 mL
5 mM	0.4068 mL	2.0339 mL	4.0679 mL	20.3393 mL
10 mM	0.2034 mL	1.0170 mL	2.0339 mL	10.1696 mL
20 mM	0.1017 mL	0.5085 mL	1.0170 mL	5.0848 mL
50 mM	0.0407 mL	0.2034 mL	0.4068 mL	2.0339 mL
100 mM	0.0203 mL	0.1017 mL	0.2034 mL	1.0170 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc