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ETRB Antagonist 1

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Catalog No. T9621Cas No. 290815-30-4

N-(6-chloro-5-(2-Methoxyphenoxy)-2-(pyridin-4-yl)pyriMidin-4-yl)-5-Met inhibits endothelin binding to membranes from CHO cells carrying human ETA receptor and human ETB receptor with IC50 of 268nM and 1810nM, respectively.

ETRB Antagonist 1

ETRB Antagonist 1

😃Good
Catalog No. T9621Cas No. 290815-30-4
N-(6-chloro-5-(2-Methoxyphenoxy)-2-(pyridin-4-yl)pyriMidin-4-yl)-5-Met inhibits endothelin binding to membranes from CHO cells carrying human ETA receptor and human ETB receptor with IC50 of 268nM and 1810nM, respectively.
Pack SizePriceAvailabilityQuantity
1 mg$148Backorder
5 mg$336Backorder
10 mg$497Backorder
25 mg$898Backorder
50 mg$1,362Backorder
100 mg$1,997Backorder
200 mg$2,994Backorder
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Product Introduction

Bioactivity
Description
N-(6-chloro-5-(2-Methoxyphenoxy)-2-(pyridin-4-yl)pyriMidin-4-yl)-5-Met inhibits endothelin binding to membranes from CHO cells carrying human ETA receptor and human ETB receptor with IC50 of 268nM and 1810nM, respectively.
Chemical Properties
Molecular Weight483.93
FormulaC22H18ClN5O4S
Cas No.290815-30-4
Relative Density.1.425 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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Keywords

N(6chloro5(2Methoxyphenoxy)2(pyridin4yl)pyriMidin4yl)5Methylpyridine2sulfonamideN (6 chloro 5 (2 Methoxyphenoxy) 2 (pyridin 4 yl)pyriMidin 4 yl) 5 Methylpyridine 2 sulfonamide
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