Powder: -20°C for 3 years | In solvent: -80°C for 1 year
6-Alpha Naloxol(Alpha-Naloxol) is an opioid antagonist and is a human metabolite of naloxone.
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Description | 6-Alpha Naloxol(Alpha-Naloxol) is an opioid antagonist and is a human metabolite of naloxone. |
In vitro | When responding over the entire 30 min operant session was examined, naloxone was only 5-fold more potent than 6-alpha-naloxol in suppressing operant responding under Morphine Na ve conditions, but this increased to a 65-fold potency difference after Single or Repeat Morphine pretreatment. Examination of the relative potency of these antagonists in the Early Phase of operant testing (5-15 min post-antagonist) revealed an even greater 100-fold potency difference between naloxone and 6-alpha-naloxol, but in the Late Phase of testing (25-35 min post-antagonist), this had declined to a 9-fold potency difference, comparable to the relative potency of naloxone to 6-alpha-naloxol under Morphine-Na ve conditions [3]. |
Synonyms | Alpha-Naloxol |
Molecular Weight | 329.39 |
Formula | C19H23NO4 |
CAS No. | 20410-95-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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6-Alpha Naloxol 20410-95-1 Others 6 Alpha Naloxol 6Alpha Naloxol Alpha-Naloxol 6-a Naloxol α-Naloxol a-Naloxol 6-α Naloxol inhibitor inhibit