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GSK4028

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Catalog No. T11495Cas No. 2079886-19-2

GSK4028 is the enantiomeric negative control of GSK4027, a PCAF/GCN5 bromodomain chemical probe, with a pIC50 of 4.9 in a TR-FRET assay.

GSK4028
Other Forms of GSK4028:
GSK 4027T11495L2079896-25-4
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GSK4028

😃Good
Catalog No. T11495Cas No. 2079886-19-2
GSK4028 is the enantiomeric negative control of GSK4027, a PCAF/GCN5 bromodomain chemical probe, with a pIC50 of 4.9 in a TR-FRET assay.
Pack SizePriceAvailabilityQuantity
5 mg$1,4708-10 weeks
10 mg$2,2008-10 weeks
25 mg$3,7408-10 weeks
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Product Introduction

Bioactivity
Description
GSK4028 is the enantiomeric negative control of GSK4027, a PCAF/GCN5 bromodomain chemical probe, with a pIC50 of 4.9 in a TR-FRET assay.
Targets&IC50
PCAF/GCN5:4.9(pIC50)
In vitro
GSK4028 also demonstrates potency toward BRD4 BD1 and BRD9 inTR-FRET assay with pIC50s of <4.3 and 4.5±0.13, respectively.GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4.9.
Chemical Properties
Molecular Weight377.28
FormulaC17H21BrN4O
Cas No.2079886-19-2
Relative Density.1.45 g/cm3 (Predicted)
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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Keywords

GSK-4028GSK 4028GSK4028
Related Tags: buy GSK4028 | purchase GSK4028 | GSK4028 cost | order GSK4028 | GSK4028 chemical structure | GSK4028 in vitro | GSK4028 formula | GSK4028 molecular weight
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