Powder: -20°C for 3 years | In solvent: -80°C for 1 year
L 888607 Racemate is a selective antagonist of prostaglandin D2 receptor subtype 1 (DP1) (Kis: 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,080.00 | |
50 mg | 6-8 weeks | $ 1,410.00 | |
100 mg | 6-8 weeks | $ 1,990.00 |
Description | L 888607 Racemate is a selective antagonist of prostaglandin D2 receptor subtype 1 (DP1) (Kis: 132 nM and 17 nM for DP1 and thromboxane A2 receptor (TP), respectively). |
Targets&IC50 | DP/DP1:132 nM (ki), TP:17 nM (ki) |
In vitro | L 888607 Racemate is actually 8-fold more effective on the TP receptor (Ki = 17 nM). L 888607 Racemate maintains a modest binding affinity for the DP1 receptor (Ki = 132 nM) . |
Molecular Weight | 375.84 |
Formula | C19H15ClFNO2S |
CAS No. | 1030017-51-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 6 mg/mL (15.96 mM), Sonification is recommended.
You can also refer to dose conversion for different animals. More
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L 888607 Racemate 1030017-51-6 Cell Cycle/Checkpoint Chromatin/Epigenetic Aurora Kinase inhibitor inhibit