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Pactimibe

Catalog No. T28290Cas No. 189198-30-9
Alias Pactimibe free base, CS-505, CS505, CS 505

Pactimibe is a ACAT inhibitor. It has anti-atherosclerotic activity.

Pactimibe
Other Forms of Pactimibe:
Pactimibe sulfateT62974608510-47-0
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Pactimibe

Catalog No. T28290Alias Pactimibe free base, CS-505, CS505, CS 505Cas No. 189198-30-9
Pactimibe is a ACAT inhibitor. It has anti-atherosclerotic activity.
Pack SizePriceAvailabilityQuantity
25 mg$1,6208-10 weeks
50 mg$2,1108-10 weeks
100 mg$3,1008-10 weeks
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Product Introduction

Bioactivity
Description
Pactimibe is a ACAT inhibitor. It has anti-atherosclerotic activity.
Targets&IC50
ACAT2:3.0 μM (IC50), ACAT:4.7 μM (IC50, in THP-1 cells), ACAT:2 μM (IC50, in the liver), Cholesteryl ester formation:6.7 μM (IC50), ACAT:2.7 μM (IC50, in macrophages), ACAT1:4.9 μM (IC50), Oleoyl-CoA:5.6 μM (Ki)
AliasPactimibe free base, CS-505, CS505, CS 505
Chemical Properties
Molecular Weight416.6
FormulaC25H40N2O3
Cas No.189198-30-9
Storage & Solubility Information
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice.

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Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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2 Enter the in vivo formulation:
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Pactimibe
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