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Pack Size | Price | Availability | Quantity |
---|---|---|---|
1 mg | $55 | In Stock | |
5 mg | $128 | In Stock | |
10 mg | $189 | In Stock | |
25 mg | $319 | In Stock | |
50 mg | $478 | In Stock | |
100 mg | $696 | In Stock | |
500 mg | $1,470 | In Stock |
Description | [DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM. [DPro10] Dynorphin A (1-11), porcine is an n-alkylated derivative with analgesic activity. |
In vitro | Porcine [DPro10] Dynorphin A (1-11) inhibits adenylyl cyclase activity in CHO cells expressing k-opioid receptors, with an IC50 value of 0.12 nM[1]. |
In vivo | Administered intracerebroventricularly (ICV), [DPro10] Dynorphin A (1-11), porcine, exhibits analgesic effects involving thermal cutaneous (tail-flick) and chemical visceral (acetic acid-induced writhing) stimuli, with known differential activation of mu and kappa receptors[2]. |
Alias | [DPro10] Dynorphin A (1-11)acetate,porcine(94596-26-6 Free base) |
Molecular Weight | 1422.7 |
Formula | C65H107N21O15 |
Cas No. |
Storage | store at low temperature,keep away from moisture Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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