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Pack Size | Price | Availability | Quantity |
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5 mg | Inquiry | Backorder | |
50 mg | Inquiry | Backorder |
Description | [DPro10] Dynorphin A (1-11), porcine hydrochloride, is an N-alkylated derivative and a potent κ-opioid receptor agonist, exhibiting a K i value of 0.13 nM. This compound possesses analgesic properties [1] [2]. |
In vitro | '[DPro10] Dynorphin A (1-11), porcine,' inhibits adenylyl cyclase activity in CHO cells expressing k-opioid receptors, exhibiting an IC50 of 0.12 nM [1]. |
In vivo | "[DPro10] Dynorphin A (1-11), porcine, administered intracerebroventricularly (ICV), exhibits analgesic properties in response to thermal cutaneous (tail-flick) and chemical visceral (AcOH-induced writhing) pain. This analgesia is mediated through the differential activation of mu and kappa opioid receptors [2]." |
Molecular Weight | 1362.62 (free acid) |
Formula | C63H103N21O13.xHCl |
Cas No. |
Storage | keep away from moisture Powder: -20°C for 3 years | In solvent: -80°C for 1 year |
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