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A2AAR antagonist 1

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Catalog No. T60591Cas No. 1784491-64-0

A2AAR antagonist 1 (compound 21a) is a potent A2AAR (adenosine A2A receptor) antagonist with high ligand efficiency and a Ki value of 20 nM. It is applicable in neurodegenerative disease research [1].

A2AAR antagonist 1

A2AAR antagonist 1

😃Good
Catalog No. T60591Cas No. 1784491-64-0
A2AAR antagonist 1 (compound 21a) is a potent A2AAR (adenosine A2A receptor) antagonist with high ligand efficiency and a Ki value of 20 nM. It is applicable in neurodegenerative disease research [1].
Pack SizePriceAvailabilityQuantity
25 mg$1,5206-8 weeks
50 mg$1,9806-8 weeks
100 mg$2,5006-8 weeks
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Product Introduction

Bioactivity
Description
A2AAR antagonist 1 (compound 21a) is a potent A2AAR (adenosine A2A receptor) antagonist with high ligand efficiency and a Ki value of 20 nM. It is applicable in neurodegenerative disease research [1].
In vitro
A2AAR antagonist 1, when applied at concentrations ranging from 0 to 10 µM for 1 hour, exhibits strong affinity for the A2AAR, evidenced by a K_i value of 20 nM [1].
Chemical Properties
Molecular Weight290.12
FormulaC12H8BrN3O
Cas No.1784491-64-0
Storage & Solubility Information
StorageShipping with blue ice.

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Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2OTargetMol | reagent mix well and clarify
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